2
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T74659 |
Dideoxy-amanitin
|
||
Dideoxy-amanitin (compound 2) 是一种α-Amanitin 衍生物,是一种强效和选择性的 RNA 聚合酶 II 变结构抑制剂,其 IC50值为 74.2 nM。 | |||
T81832 |
MC-VC-PABC-C6-alpha-Amanitin
|
||
MC-VC-PABC-C6-alpha-Amanitin是一款针对HER2受体的ADC,包含致癌毒素alpha-Amanitin及单克隆抗体MC-VC-PABC-C6。alpha-Amanitin主要抑制RNA聚合酶IIα。该化合物专一性地靶向HER2阳性肿瘤细胞,主要应用于乳腺癌与胃癌的研究领域。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T39649 |
ε-Amanitin
|
||
ε-Amanitin is a cyclic peptide obtained from various mushroom species. It exhibits a strong affinity for RNA polymerase II and effectively inhibits its activity. | |||
T39562 |
γ-Amanitin
|
||
γ-Amanitin an ADC cytotoxin and isolated from the mushroom. γ-Amanitin inhibits RNA polymerase II and disrupts synthesis of mRNA. γ-Amanitin shows similar effects to α-Amanitin and β-Amanitin. |