Cat. No. | Product Name | Target | Signaling Pathways |
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TP1892 |
γ1-MSH
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Endogenous melanocortin MC3 receptor agonist (pKi = 7.46) that displays ~ 40-fold selectivity over MC4. Increases the release of extracellular dopamine, which induces grooming and vertical activity (rearing) in rats. Exhibits hypertensive, tachycardic and | |||
T75851 |
γ1-MSH TFA
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γ1-MSH TFA 是黑素皮质素 MC3受体激动剂,对大鼠 MC3受体的 Ki 为 34 nM。γ1-MSH TFA 在 MC4 (Ki=1318 nM) 上表现出约 40 倍的选择性。 | |||
TP1002L |
γ-1-MSH, amide acetate (72629-65-3 free base)
γ-1-MSH, amide acetate |
Others | Others |
γ-1-MSH, amide acetate (72629-65-3 free base) 是 ACTH/β-内啡肽 (β-EP) 前体蛋白 N 末端区域的一种推定激素,RIA 使用抗 γ-3-MSH 抗血清对产生 ACTH 的小鼠进行了研究垂体肿瘤细胞,AtT-20/D16v。 | |||
T75971 |
γ-1-Melanocyte Stimulating Hormone (MSH), amide
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γ-1-Melanocyte Stimulating Hormone (MSH), amide为含11个氨基酸的多肽,主要通过激活黑皮质素受体3 (MC3-R) 调节钠 (Na+) 平衡及血压。 |