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Cat. No. Product Name Target Signaling Pathways
TP1369L [Sar9,Met(O2)11]-Substance P acetate

[Sar9,Met(O2)11]-Substance P acetate(110880-55-2 free base)

Neurokinin receptor GPCR/G Protein; Neuroscience
[Sar9,Met(O2)11]-Substance P acetate(110880-55-2 free base) 是一种速激肽 NK1 受体选择性激动剂。它是一种选择性速激肽 NK1 受体激动剂。它和 septide(每只大鼠 10-100 pmol,i.c.v.)在增加平均动脉血压 (MAP) 和心率 (HR),但它们的时间进程不同。两种激动剂都以剂量依赖性方式增加洗脸和吸鼻,而它是一种产生美容效果的化合物。
T7828 [Sar9,Met(O2)11]-Substance P

Bhsar-sp,NA,精氨酰-脯氨酰-赖氨酰-脯氨酰-谷氨酰-谷氨酰-苯丙氨酰-苯丙氨酰-SAR-亮氨酸-蛋氨酸[O2]-胺

Neurokinin receptor GPCR/G Protein; Neuroscience
[Sar9,Met(O2)11]-Substance P (NA) 是选择性速激肽NK1受体激动剂。
TP1369 [Sar9,Met(O2)11]-Substance P TFA(110880-55-2,free)

[Sar9,Met(O2)11]-Substance P TFA

[Sar9,Met(O2)11]-Substance P TFA is a selective tachykinin NK1 receptor agonist.[Sar9,Met(O2)11]-Substance P and septide (10-100 pmol per rat, i.c.v.) are equipotent in increasing mean arterial blood pressure (MAP) and heart rate (HR), yet they have dissi
T75769 [Sar9,Met(O2)11]-Substance P TFA

[Sar9,Met(O2)11]-Substance P TFA 是一种选择性的速激肽NK1受体激动剂。
TP1862L [Sar9] Substance P acetate(77128-75-7 free base)

Neurokinin receptor GPCR/G Protein; Neuroscience
[Sar9] Substance P acetate(77128-75-7 free base) 是一种 NK-1 受体激动剂。 rNK1 特异性激动剂 [Sar-9,Met(O2)11]-SP 模拟了 SP 对孕酮代谢的作用。
T70456 Nolpitantium Free Base

Nolpitantium Free Base is a highly selective nonpeptide antagonist of neurokinin-1 (NK1) receptor. Nolpitantium potently, selectively and competitively inhibited substance P binding to NK1 receptors from various animal species, including humans. In vitro, it was a potent antagonist in functional assays for NK1 receptors such as [Sar9, Met(O2)11]substance P-induced endothelium-dependent relaxation of rabbit pulmonary artery and contraction of guinea-pig ileum. Up to 1 mkM, Nolpitantium had no eff...
TP1862 [Sar9] Substance P

[Sar9]-Substance P is one of NK-1 receptor agonist. The action of SP on progesterone metabolism was mimicked by the rNK1-specific agonist [Sar-9,Met(O2)11]-SP.

化合物

[Sar9,Met(O2)11]-Substance P acetate
Cat.No: TP1369L
Synonym: [Sar9,Met(O2)11]-Substance P acetate(110880-55-2 free base)
Target: Neurokinin receptor
[Sar9,Met(O2)11]-Substance P
Cat.No: T7828
Synonym: Bhsar-sp,NA,精氨酰-脯氨酰-赖氨酰-脯氨酰-谷氨酰-谷氨酰-苯丙氨酰-苯丙氨酰-SAR-亮氨酸-蛋氨酸[O2]-胺
Target: Neurokinin receptor
[Sar9,Met(O2)11]-Substance P TFA(110880-55-2,free)
Cat.No: TP1369
Synonym: [Sar9,Met(O2)11]-Substance P TFA
Target:
[Sar9,Met(O2)11]-Substance P TFA
Cat.No: T75769
Synonym:
Target:
[Sar9] Substance P acetate(77128-75-7 free base)
Cat.No: TP1862L
Synonym:
Target: Neurokinin receptor
Nolpitantium Free Base
Cat.No: T70456
Synonym:
Target:
[Sar9] Substance P
Cat.No: TP1862
Synonym:
Target:
TargetMol Loading
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