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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T125054 Variabilin

化合物

Variabilin
Cat.No: T125054
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN5221 (-)-Variabilin

Variabilin, a novel inhibitor of human platelet aggregation, it is a potent RGD (Arg-Gly-Asp)-containing antagonist of the fibrinogen receptor glycoprotein IIb-IIIa (GPIIb-IIIa; αIIbβ3) and the vitronectin receptor αvβ3.Variabilin is also an antimicrobial furanosesterterpene. Variabilin is an inhibitor of human secretory and cytosolic phospholipase A2 (PLA2) activities that controls eicosanoid production in vitro and in vivo, inhibits neutrophil degranulation and superoxide generation in vitro a...

天然产物

(-)-Variabilin
Cat.No: TN5221
Synonym:
Target:
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