ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1835 | Ibrutinib | 936563-96-1 | 440.5 | 10mM | BTK; Ligands for Target Protein for PROTAC; Src; Tyrosine Kinases |
T1976 | RN486 | 1242156-23-5 | 606.69 | 10mM | BTK |
T2302 | CNX-774 | 1202759-32-7 | 499.5 | 10mM | BTK |
T2472 | CGI-1746 | 910232-84-7 | 579.69 | 10mM | Autophagy; BTK |
T3024 | Avitinib | 1557267-42-1 | 487.53 | 10mM | BTK; EGFR; JAK |
T3626 | Acalabrutinib | 1420477-60-6 | 465.51 | 10mM | BTK |
T4268 | CHMFL-BMX-078 | 1808288-51-8 | 625.67 | 10mM | BTK |
T4337 | PCI 29732 | 330786-25-9 | 371.44 | 10mM | BCRP; BTK |
T4387 | evobrutinib | 1415823-73-2 | 429.52 | 10mM | BTK |
T6078 | Saracatinib | 379231-04-6 | 542.03 | 10mM | Autophagy; BTK; EGFR; Src |
T6217 | LFM-A13 | 244240-24-2 | 360.01 | 10mM | BTK; JAK; PLK |
T6918 | Olmutinib | 1353550-13-6 | 486.59 | 10mM | BTK; EGFR |
T6921 | ONO-4059 analog | 1351635-67-0 | 456.5 | 10mM | Apoptosis; BTK |
T5138 | BMS-986142 | 1643368-58-4 | 572.6 | 10mM | BTK |
T5407 | Branebrutinib | 1912445-55-6 | 370.43 | 10mM | BTK |
T7584 | zanubrutinib | 1691249-45-2 | 471.55 | 10mM | BTK |
T12317 | Orelabrutinib | 1655504-04-3 | 427.5 | 10mM | BTK |
T12542 | Rilzabrutinib | 1575596-29-0 | 665.76 | 10mM | BTK; EGFR; HER |
T14323 | ARQ 531 | 2095393-15-8 | 478.93 | 10mM | BTK |
T10629 | Btk inhibitor 2 | 1558036-85-3 | 431.49 | 10mM | BTK |
TQ0230 | BTK IN-1 | 1270014-40-8 | 384.86 | 10mM | BTK |
T16730 | Remibrutinib | 1787294-07-8 | 507.53 | 10mM | BTK |
TQ0242 | Fenebrutinib | 1434048-34-6 | 664.8 | 10mM | BTK |
T9072 | Tuxobertinib | 2414572-47-5 | 561.03 | 10mM | BTK; EGFR; HER; RIP kinase |
T9125 | Tolebrutinib | 1971920-73-6 | 455.51 | 10mM | BTK |
T9192 | BIIB068 | 1798787-27-5 | 435.52 | 10mM | BTK |
T12311 | Tirabrutinib hydrochloride | 1439901-97-9 | 490.94 | 10mM | BTK |
T13564 | AZ7550 | 1421373-99-0 | 485.58 | 10mM | ACK; ALK; BTK; Drug Metabolite; EGFR; FAK; FLT; IGF-1R; MLK; MNK; PYK2; Tyrosine Kinases |
T9408 | N-piperidine Ibrutinib | 330785-90-5 | 386.45 | 10mM | BTK |
T16157 | MT-802 | 2231744-29-7 | 787.82 | 10mM | BTK; PROTACs |
T9705 | TL-895 | 1415823-49-2 | 447.5 | 10mM | BTK |
T36287 | Pirtobrutinib | 2101700-15-4 | 479.43 | 10mM | BTK |
T14692 | BMX-IN-1 | 1431525-23-3 | 524.59 | 10mM | BTK |
T17098 | Tilfrinib | 1600515-49-8 | 275.3 | 10mM | BTK |