BET inhibitor kit 包含 BET 抑制剂,BET 抑制剂通过模拟乙酰化的 Lys 结构与 KAc 口袋结合,阻断 BD1或 BD2与 KAc 结合,从而在表观遗传学水平上对基因表达进行调控,可用于白血病、淋巴瘤、乳腺癌、脑瘤和骨髓瘤等的治疗研究。TargetMol 为您提供47种精选BET 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1854 | MS436 | 1395084-25-9 | 383.42 | 10mM | Epigenetic Reader Domain |
T1906 | Molibresib | 1260907-17-2 | 423.9 | 10mM | Epigenetic Reader Domain |
T2072 | BET bromodomain inhibitor | 1505453-59-7 | 445.91 | 10mM | Epigenetic Reader Domain |
T2091 | CPI0610 | 1380087-89-7 | 365.81 | 10mM | c-Myc; Epigenetic Reader Domain |
T2110 | (+)-JQ-1 | 1268524-70-4 | 456.99 | 10mM | Autophagy; Epigenetic Reader Domain; Ligands for Target Protein for PROTAC |
T2120 | I-BET151 | 1300031-49-5 | 415.44 | 10mM | Epigenetic Reader Domain |
T2480 | Apabetalone | 1044870-39-4 | 370.4 | 10mM | Epigenetic Reader Domain; HIV Protease |
T3504 | AZD5153 6-Hydroxy-2-naphthoic acid | 1869912-40-2 | 667.75 | 10mM | Epigenetic Reader Domain |
T3712 | Mivebresib | 1445993-26-9 | 459.47 | 10mM | Apoptosis; Epigenetic Reader Domain |
T4247 | I-CBP112 hydrochloride | 2147701-33-3 | 505 | 10mM | Epigenetic Reader Domain |
T4345 | CeMMEC1 | 440662-09-9 | 336.35 | 10mM | Carboxypeptidase; DNA/RNA Synthesis; Epigenetic Reader Domain |
T4365 | FL-411 | 2118944-88-8 | 341.43 | 10mM | Epigenetic Reader Domain |
T6021 | GSK1324726A | 1300031-52-0 | 434.91 | 10mM | Apoptosis; Epigenetic Reader Domain |
T6032 | Birabresib | 202590-98-5 | 491.99 | 10mM | Epigenetic Reader Domain |
T6173 | BI 2536 | 755038-02-9 | 521.66 | 10mM | Apoptosis; Epigenetic Reader Domain; PLK |
T6222 | PFI-1 | 1403764-72-6 | 347.39 | 10mM | Apoptosis; Autophagy; Epigenetic Reader Domain |
T5362 | Y06036 | 1832671-96-1 | 427.27 | 10mM | Epigenetic Reader Domain |
T5417 | INCB-057643 | 1820889-23-3 | 415.46 | 10mM | Apoptosis; Epigenetic Reader Domain |
T6828 | ZL0420 | 2229039-45-4 | 296.32 | 10mM | Epigenetic Reader Domain |
T7863 | Hexamethylene bisacetamide | 3073-59-4 | 200.28 | 10mM | Epigenetic Reader Domain |
T8495 | Alobresib | 1637771-14-2 | 437.5 | 10mM | Epigenetic Reader Domain |
T19618 | (R)-(-)-JQ1 Enantiomer | 1268524-71-5 | 456.99 | 10mM | Epigenetic Reader Domain |
T17311 | (+)-JQ1 PA | 2115701-93-2 | 437.95 | 10mM | Epigenetic Reader Domain |
TQ0253 | PLX51107 | 1627929-55-8 | 438.48 | 10mM | Epigenetic Reader Domain |
T16154 | MS417 | 916489-36-6 | 414.91 | 10mM | Epigenetic Reader Domain; HIV Protease |
T8601 | 1-benzyl-2-ethyl-4,5,6,7-tetrahydro-1H-indol-4-one | 218934-50-0 | 253.35 | 10mM | Epigenetic Reader Domain |
T8609 | CHEMBRDG-BB 7118966 | 328956-24-7 | 241.09 | 10mM | Epigenetic Reader Domain |
T8658 | NEO2734 | 2081072-29-7 | 435.44 | 10mM | Epigenetic Reader Domain; Histone Acetyltransferase |
T19935 | XD14 | 1370888-71-3 | 421.51 | 10mM | Epigenetic Reader Domain |
T12112 | MS402 | 1672684-68-2 | 370.83 | 10mM | Epigenetic Reader Domain |
T8932 | GSK046 | 2474876-09-8 | 414.48 | 10mM | Epigenetic Reader Domain |
T9020 | GSK620 | 2088410-46-0 | 325.4 | 10mM | Epigenetic Reader Domain |
T9194 | UMB298 | 2266569-73-5 | 479.01 | 10mM | Epigenetic Reader Domain |
T50006 | 3-methyl-1,2,3,4-tetrahydroquinazolin-2-one | 24365-65-9 | 162.19 | 10mM | Epigenetic Reader Domain |
T14776 | BRD4 Inhibitor-10 | 1660117-38-3 | 429.51 | 10mM | Epigenetic Reader Domain |
T15405 | GNE-781 | 1936422-33-1 | 525.59 | 10mM | Epigenetic Reader Domain |
T10521 | ODM-207 | 1801503-93-4 | 375.42 | 10mM | Epigenetic Reader Domain |
T28628 | RVX-297 | 1044871-04-6 | 423.5 | 10mM | Epigenetic Reader Domain |
T9629 | WAY-309060 | 309951-18-6 | 262.26 | 10mM | Epigenetic Reader Domain |
T9703L | GSK778 hydrochloride | T9703L | 548.08 | 10mM | Epigenetic Reader Domain |
T13363 | Y06137 | 2226534-49-0 | 444.57 | 10mM | Epigenetic Reader Domain |
T60072 | ZL0590 | 2230496-99-6 | 512.55 | 10mM | Epigenetic Reader Domain |
T22345 | INCB054329 | 1628607-64-6 | 348.36 | 10mM | Epigenetic Reader Domain; Others |
T13394 | ZEN-3862 | 1952264-33-3 | 340.35 | 10mM | Epigenetic Reader Domain |
T27392 | FT001 | 1778655-51-8 | 467.58 | 10mM | Epigenetic Reader Domain |
T12338 | OXFBD04 | 2231747-03-6 | 296.32 | 10mM | Epigenetic Reader Domain |
T12513 | PNZ5 | 1629277-36-6 | 318.37 | 10mM | Epigenetic Reader Domain |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |