Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Caroverine hydrochloride (Caroverine HCL) 是竞争性可逆的NMDA 和AMPA 谷氨酸受体拮抗剂。它也是抗氧化和钙阻滞剂,具有血管舒张作用,可用于内耳耳鸣的研究。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 185 | 现货 | ||
5 mg | ¥ 413 | 现货 | ||
10 mg | ¥ 663 | 现货 | ||
25 mg | ¥ 1,370 | 现货 | ||
50 mg | ¥ 2,320 | 现货 | ||
100 mg | ¥ 3,930 | 现货 | ||
200 mg | ¥ 5,630 | 现货 | ||
500 mg | ¥ 8,490 | 现货 | ||
1 mL * 10 mM (in DMSO) | ¥ 455 | 现货 |
产品描述 | Caroverine hydrochloride (Caroverine HCL) is a potent, competitive and reversible antagonist of NMDA and AMPA glutamate receptor. It is also an antioxidant and calcium-blocking agent that exhibits vasorelaxant action, and can be used for the research of inner ear tinnitus. |
体内活性 | Caroverine (1 μM; pretreated for 10 min) inhibits the pressor response to KCl (80 mM) and noradrenaline (1 μM) in the rat hindquarter preparation. Caroverine markedly suppresses the contraction caused by KCl (40 mM) in the rat isolated aorta[1].Caroverine (1.44 mg/rat; s.c; 1.0 mL/h for 72 h) attenuates impulse noise-induced hearing loss in the rat[2] |
别名 | Caroverine HCL |
分子量 | 401.9 |
分子式 | C22H28ClN3O2 |
CAS No. | 55750-05-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (248.80 mM), sonification is recommended.
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 2.4882 mL | 12.4409 mL | 24.8818 mL | 62.2045 mL |
5 mM | 0.4976 mL | 2.4882 mL | 4.9764 mL | 12.4409 mL | |
10 mM | 0.2488 mL | 1.2441 mL | 2.4882 mL | 6.2205 mL | |
20 mM | 0.1244 mL | 0.622 mL | 1.2441 mL | 3.1102 mL | |
50 mM | 0.0498 mL | 0.2488 mL | 0.4976 mL | 1.2441 mL | |
100 mM | 0.0249 mL | 0.1244 mL | 0.2488 mL | 0.622 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
Caroverine hydrochloride 55750-05-5 Membrane transporter/Ion channel Neuroscience GluR NMDAR iGluR NMDA glutamate calcium Tinnex tinnitus vasorelaxant antioxidant Caroverine Hydrochloride Inhibitor inner inhibit ear Caroverine HCL Ionotropic glutamate receptors AMPA Caroverine inhibitor