Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 1,055 | 待询 | ||
2 mg | ¥ 1,735 | 待询 | ||
5 mg | ¥ 3,010 | 待询 | ||
10 mg | ¥ 4,710 | 待询 | ||
25 mg | ¥ 8,450 | 待询 | ||
50 mg | ¥ 14,060 | 待询 | ||
100 mg | ¥ 19,160 | 待询 | ||
200 mg | 待询 | 待询 | ||
500 mg | 待询 | 待询 | ||
1 mL * 10 mM (in DMSO) | ¥ 3,235 | 待询 |
产品描述 | GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM). |
靶点活性 | GRK2:30 nM, GRK5:7.1 μM |
体外活性 | GRKs-IN-1 hydrochloride (Compound 14as) is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine. |
别名 | GRK2-IN-1 hydrochloride |
分子量 | 488.94 |
分子式 | C24H26ClFN4O4 |
CAS No. | T13714L |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 250 mg/mL (511.31 mM), sonification is recommended.
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 2.0452 mL | 10.2262 mL | 20.4524 mL | 51.131 mL |
5 mM | 0.409 mL | 2.0452 mL | 4.0905 mL | 10.2262 mL | |
10 mM | 0.2045 mL | 1.0226 mL | 2.0452 mL | 5.1131 mL | |
20 mM | 0.1023 mL | 0.5113 mL | 1.0226 mL | 2.5566 mL | |
50 mM | 0.0409 mL | 0.2045 mL | 0.409 mL | 1.0226 mL | |
100 mM | 0.0205 mL | 0.1023 mL | 0.2045 mL | 0.5113 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
GRK2-IN-1 hydrochloride (2055990-90-2 free base) T13714L GPCR/G Protein GRK GRK2-IN-1 Hydrochloride 2055990-90-2 GRK-2-IN-1 hydrochloride (2055990-90-2 free base) GRK2IN1 hydrochloride (2055990902 free base) GRK2-IN-1 hydrochloride 2055990-90-2 free base GRK2 IN 1 hydrochloride (2055990 90 2 free base) Inhibitor inhibitor inhibit