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TargetMol | Compound Library

抗前列腺癌化合物库现货

Anti-Prostate Cancer Compound Library

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产品编号 L2195

前列腺癌是指发生在前列腺的上皮性恶性肿瘤,是男性生殖系统中常见的恶性肿瘤,具有复杂的疾病发病机制。Androgen Receptor、Hedgehog、TGF-β、Wnt、PI3K-AKT-mTOR 等多个信号通路和靶点参与前列腺癌的进展。 TargetMol 抗前列腺癌化合物库收集了2256 种与前列腺癌相关的化合物,包括已经报道具有前列腺癌治疗作用的化合物,以及靶向前列腺癌相关靶点的化合物,是抗前列腺癌药物研发的良好工具。

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产品编号 L2195

抗前列腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2256种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
VEGFR
EGFR
Reactive Oxygen Species
COX
mTOR
ERK
Akt
PARP
CDK
Wnt/beta-catenin
JAK
Endogenous Metabolite
AMPK
p38 MAPK
GSK-3
STAT
FGFR
Androgen Receptor
PDGFR
Antibacterial
Raf
MEK
Src
Ras
FLT
c-Kit
JNK
MAPK
IκB/IKK
TNF
DNA-PK
Histone Methyltransferase
S6 Kinase
Caspase
Parasite
Hedgehog/Smoothened
ATM/ATR
Cytochromes P450
Tyrosine Kinases
IL Receptor
Potassium Channel
Antifungal
Ferroptosis
c-Met/HGFR
PPAR
RIP kinase
PDK
Antibiotic
HER
Pim
Aurora Kinase
c-RET
NOD
HIV Protease
Antioxidant
Bcr-Abl
Influenza Virus
PKC
Mitophagy
Gamma-secretase
Epigenetic Reader Domain
NO Synthase
Calcium Channel
Casein Kinase
PKA
IRAK
PD-1/PD-L1
Estrogen/progestogen Receptor
Rho
ROS
MMP
IGF-1R
Bcl-2 Family
PI4K
Lipoxygenase
DNA/RNA Synthesis
Microtubule Associated
Smo
Nrf2
NOD-like Receptor (NLR)
p53
Dehydrogenase
Virus Protease
Topoisomerase
Mitochondrial Metabolism
c-Fms
HDAC
NOS
Prostaglandin Receptor
GABA Receptor
Estrogen Receptor/ERR
Chk
TGF-beta/Smad
Beta Amyloid
AChR
Tyrosinase
HIF/HIF Prolyl-Hydroxylase
Phosphatase
ROCK
PDE
Interleukin
Trk receptor
Syk
Sodium Channel
FAK
Kras
GNRH Receptor
SIK
E1/E2/E3 Enzyme
Drug Metabolite
PTEN
P-gp
TLR
5-HT Receptor
PLK
Proteasome
DYRK
NADPH
Adrenergic Receptor
CSF-1R
Antifection
HSV
Cholinesterase (ChE)
PGE Synthase
Antiviral
HSP
MELK
TAM Receptor
Carbonic Anhydrase
Transferase
HCV Protease
Integrin
RAAS
Tie-2
HBV
TRP/TRPV Channel
Glucocorticoid Receptor
MNK
SARS-CoV
Ephrin Receptor
ASK
HIF
Reductase
Histamine Receptor
Glutathione Peroxidase
TOPK
Progesterone Receptor
Serine Protease
Aryl Hydrocarbon Receptor
IAP
LDL
Glucosidase
Opioid Receptor
Porcupine
Free radical scavengers
Histone Acetyltransferase
transporter
ALK
SGK
Cannabinoid Receptor
Anti-infection
MLK
GPCR
Mdm2
ATPase
Chloride channel
IFNAR
BACE
GTPase
c-Myc
Cholecystokinin Receptor
Leukotriene Receptor
IRE1
Fatty Acid Synthase
CXCR
CaMK
PSMA
Hippo pathway
Retinoid Receptor
KLF
Phospholipase
BTK
RAR/RXR
Dopamine Receptor
ROR
ADC Cytotoxin
YAP
Adenosine Receptor
PERK
MRP
Serine/threonin kinase
RANKL/RANK
MAO
NMDAR
ABC Transporter
DNA Alkylation
FAAH
CCR
Endothelin Receptor
cAMP
GluR
DUB
Beta-Secretase
Acyltransferase
STING
LRRK2
Reverse Transcriptase
Discoidin Domain Receptor (DDR)
Gap Junction Protein
NADPH-oxidase
S1P Receptor
Melanin-concentrating Hormone Receptor (MCHR)
Apelin receptor
Proton pump
MicroRNA
NPC1L1
DHFR
Arginase
LTR
Na+/Ca2+ Exchanger
gp120/CD4
VDA
OCT
Hck
Nucleoside Antimetabolite/Analog
Cysteine Protease
Liver X Receptor
FXR
Glucokinase
PYK2
iGluR
Myosin
FLAP
UGT
PAFR
Haspin Kinase
Monoamine Transporter
DPP-4
PAK
ACK1
Somatostatin
DNA
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Wee1
ATP Citrate Lyase
BCRP
OXPHOS
Glutathione reductase
Survivin
Aminopeptidase
Sirtuin
CD73
Decarboxylase
cGAS
hCE
PAI-1
RSV
Methionine Adenosyltransferase (MAT)
GST
GPX
Aromatase
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
DAPK
Platelet aggregation
BMI-1
DNA Methyltransferase
Sigma receptor
AhR
CFTR
PKM
Kinesin
Monoamine Oxidase

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