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HIV Protease

HIV Protease

HIV-1 protease (PR) is a retroviral aspartyl protease (retropepsin), an enzyme involved with peptide bond hydrolysis in retroviruses, that is essential for the life-cycle of HIV, the retrovirus that causes AIDS. HIV protease cleaves newly synthesized polyproteins (namely, Gag and Gag-Pol[3]) at nine cleavage sites to create the mature protein components of an HIV virion, the infectious form of a virus outside of the host cell. Without effective HIV protease, HIV virions remain uninfectious.
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Cat. No. Product Name CAS No. Purity Chemical Structure
T16112 ML67-33
化合物 T16112
1443290-89-8 98%
ML67-33 rapidly and reversibly affects K2P2.1 (TREK-1) (EC50s: 36.3 μM and 9.7 μM in cell-free and HEK293 cells, respectively). ML67-33 is a selective activator ...
TN1670 Ganodermanondiol
灵芝酮二醇
107900-76-5 98%
Ganodermanondiol exhibits potent cytoprotective effects on t-BHP-induced hepatotoxicity in human liver-derived HepG2 cells, presumably through Nrf2-mediated anti...
T12420 Pentosan Polysulfate
化合物 T12420
37300-21-3 98%
Pentosan Polysulfate is a potent and selective anti-HIV agent.with anti-inflammatory and pro-chondrogenic properties,and used for treatment of interstitial cysti...
TN4911 Rhuscholide A
化合物 TN4911
944804-58-4 98%
Rhuscholide A possesses significant anti-HIV-1 activity with an EC50 value of 1.62 microM and a therapeutic index (TI) of 42.40.
TN5012 Shizukaol C
化合物 TN5012
142279-41-2 98%
1. Shizukaol C shows anti-HIV-1 replication activities in both wild-type HIV-1 and two NNRTIs-resistant strains.
2. Shizukaol C has significant cytotoxicit...
T16555 PNU-103017
化合物 T16555
166335-18-8 98%
PNU-103017 is an inhibitor of HIV protease.
TN1302 6,8-Diprenylorobol
化合物6,8-Diprenylorobol
66777-70-6 98%
6,8-Diprenylorobol possesses weaker anti-H. pylori activity, it may be a useful chemopreventive agent for peptic ulcer or gastric cancer in H. pylori-infected in...
TN4264 Isoapetalic acid
化合物 TN4264
34366-34-2 98%
Isoapetalic acid and apetalic acid exhibit cytotoxic activities towards both cancer cell lines(human breast cancer (MCF-7) and human lung carcinoma (A-549) cell ...
T39264L Cyclotriazadisulfonamide hydrochloride
化合物 Cyclotriazadisulfonamide hydrochloride
392287-03-5 98%
Cyclotriazadisulfonamide hydrochloride 是 CD4 靶向 HIV 进入的选择性抑制剂,并以信号肽依赖性方式抑制人 CD4 共翻译易位进入 ER 腔。
TN1852 Lancifodilactone F
化合物 TN1852
850878-47-6 98%
Lancifodilactone F exerts minimal cytotoxicity against C8166 cells (CC50 > 200 microg/mL) and shows anti-HIV activity with EC50 = 20.69 +/- 3.31 microg/mL and a ...
TN4835 Przewalskin
化合物 TN4835
119400-87-2 98%
Przewalskin A and Przewalskin B showed modest anti-HIV-1 activity with EC50 = 41 and 30 microg/mL, respectively.
TN1660 Ganoderic acid C1
灵芝酸C1
95311-97-0 98%
Ganoderic acid C1 是分离自 G. lucidum 中的天然产物,能够抑制小鼠巨噬细胞TNF-α 的生成。
T10714 CCR5 antagonist 1
化合物 T10714
716354-86-8 98%
CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.
T30791 Censavudine
化合物Censavudine
634907-30-5 98%
Censavudine (OBP-601) 是一种核苷类似物,是一种核苷逆转录酶 (nucleoside reverse transcriptase) 抑制剂,可用于预防和治疗人类免疫缺陷病毒 1 (HIV-1)。Censavudine 对 HIV-2 和 HIV-1 具有抑制作用, EC50 范围分别为 30-81 n...
TMA1012 Ganoderiol F
化合物 TMA1012
114567-47-4 98%
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
T12420L Pentosan Polysulfate Sodium (W/W 43%)
化合物 T12420L
140207-93-8 98%
Pentosan Polysulfate Sodium is a potent and selective anti-HIV agent.with anti-inflammatory and pro-chondrogenic properties,and used for treatment of interstitia...
TN4934 Salaspermic acid
化合物 TN4934
71247-78-4 98%
Salaspermic acid is an inhibitor of HIV reverse transcriptase and HIV replication in H9 lymphocyte cells.
T13796 Nigranoic acid
化合物 T13796
39111-07-4 98%
Nigranoic acid is a natural product,and inhibits HIV-1 reverse transcriptase.
TQ0073 Andropanolide
穿心莲内酯
869807-57-8 98%
Andropanolide 是一种来自穿心莲的二帖类化合物,具有抗HIV、抗疟和抗癌活性,对 Lipopolysaccharides (LPS) 刺激的 RAW264.7 巨噬细胞中一氧化氮 (NO) 的过量产生有抑制作用。
TN3444 Aristolactam BII
化合物 TN3444
53948-09-7 98%
Aristolactam BII exhibits antimicrobial and antiinflammatory activity, it shows significant activity towards DPPH radical scavenging and potent inhibitory effect...
ML67-33
T16112
ML67-33 rapidly and reversibly affects K2P2.1 (TREK-1) (EC50s: 36.3 μM and 9.7 μM in cell-free and HEK293 cells, respectively). ML67-33 is a selective activator ...
Ganodermanondiol
TN1670
Ganodermanondiol exhibits potent cytoprotective effects on t-BHP-induced hepatotoxicity in human liver-derived HepG2 cells, presumably through Nrf2-mediated anti...
Pentosan Polysulfate
T12420
Pentosan Polysulfate is a potent and selective anti-HIV agent.with anti-inflammatory and pro-chondrogenic properties,and used for treatment of interstitial cysti...
Rhuscholide A
TN4911
Rhuscholide A possesses significant anti-HIV-1 activity with an EC50 value of 1.62 microM and a therapeutic index (TI) of 42.40.
Shizukaol C
TN5012
1. Shizukaol C shows anti-HIV-1 replication activities in both wild-type HIV-1 and two NNRTIs-resistant strains. <br/> 2. Shizukaol C has significant cytotoxicit...
PNU-103017
T16555
PNU-103017 is an inhibitor of HIV protease.
6,8-Diprenylorobol
TN1302
6,8-Diprenylorobol possesses weaker anti-H. pylori activity, it may be a useful chemopreventive agent for peptic ulcer or gastric cancer in H. pylori-infected in...
Isoapetalic acid
TN4264
Isoapetalic acid and apetalic acid exhibit cytotoxic activities towards both cancer cell lines(human breast cancer (MCF-7) and human lung carcinoma (A-549) cell ...
Cyclotriazadisulfonamide hydrochloride
T39264L
Cyclotriazadisulfonamide hydrochloride 是 CD4 靶向 HIV 进入的选择性抑制剂,并以信号肽依赖性方式抑制人 CD4 共翻译易位进入 ER 腔。
Lancifodilactone F
TN1852
Lancifodilactone F exerts minimal cytotoxicity against C8166 cells (CC50 > 200 microg/mL) and shows anti-HIV activity with EC50 = 20.69 +/- 3.31 microg/mL and a ...
Przewalskin
TN4835
Przewalskin A and Przewalskin B showed modest anti-HIV-1 activity with EC50 = 41 and 30 microg/mL, respectively.
Ganoderic acid C1
TN1660
Ganoderic acid C1 是分离自 G. lucidum 中的天然产物,能够抑制小鼠巨噬细胞TNF-α 的生成。
CCR5 antagonist 1
T10714
CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.
Censavudine
T30791
Censavudine (OBP-601) 是一种核苷类似物,是一种核苷逆转录酶 (nucleoside reverse transcriptase) 抑制剂,可用于预防和治疗人类免疫缺陷病毒 1 (HIV-1)。Censavudine 对 HIV-2 和 HIV-1 具有抑制作用, EC50 范围分别为 30-81 n...
Ganoderiol F
TMA1012
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
Pentosan Polysulfate Sodium (W/W 43%)
T12420L
Pentosan Polysulfate Sodium is a potent and selective anti-HIV agent.with anti-inflammatory and pro-chondrogenic properties,and used for treatment of interstitia...
Salaspermic acid
TN4934
Salaspermic acid is an inhibitor of HIV reverse transcriptase and HIV replication in H9 lymphocyte cells.
Nigranoic acid
T13796
Nigranoic acid is a natural product,and inhibits HIV-1 reverse transcriptase.
Andropanolide
TQ0073
Andropanolide 是一种来自穿心莲的二帖类化合物,具有抗HIV、抗疟和抗癌活性,对 Lipopolysaccharides (LPS) 刺激的 RAW264.7 巨噬细胞中一氧化氮 (NO) 的过量产生有抑制作用。
Aristolactam BII
TN3444
Aristolactam BII exhibits antimicrobial and antiinflammatory activity, it shows significant activity towards DPPH radical scavenging and potent inhibitory effect...
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