Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product Name	CAS No.	Purity
TCS2185	Yohimbine 育亨宾	146-48-5
TCS2185	Yohimbine 是一种有效的、相对非选择性的α2 - 肾上腺素能受体拮抗剂，IC50=0.6μM。
T1769	Pardoprunox 帕多芦诺	269718-84-5
T1769	Pardoprunox (SLV-308) 是多巴胺受体D2、D3部分激动剂和5-HT1A 激动剂，pEC50分别为 8、9.2 和 6.3。
TN4882	Quinine HCl 化合物 TN4882	130-89-2	98%
TN4882	Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T5450	DL-071-IT 化合物DL-071-IT	55104-39-7	98%
T5450	DL-071-IT (Afurolol Hydrochloride) 是一种有效的非选择性β-肾上腺素受体拮抗剂。 DL-071-IT 表现出内在的拟交感神经活性和弱的膜稳定活性。
T13470	(±)-Levomepromazine-d6 化合物 T13470	1189805-51-3	98%
T13470	(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T78567	Moprolol 化合物 Moprolol	5741-22-0	98%
T78567	Moprolol ((±)-Moprolol)为β-肾上腺素能受体阻滞剂，主要应用于原发性高血压研究。
T79641	(±)-N-Methylcoclaurine 化合物 (±)-N-Methylcoclaurine	1472-62-4	98%
T79641	(±)-N-Methylcoclaurine为选择性α2-肾上腺素受体拮抗剂。
T80175	Conopeptide rho-TIA 化合物 Conopeptide rho-TIA	381725-58-2	98%
T80175	Conopeptide rho-TIA为从掠食性海螺Conus tulipa毒液中提炼的多肽，对人类α1B-Adrenergic Receptor呈现非竞争性抑制作用，同时对α1A-Adrenergic Receptor和α1D-Adrenergic Receptor表现出竞争性抑制。Conopeptide rho-TI...
T80477	Muscarinic toxin 3 化合物 Muscarinic toxin 3	873336-87-9	98%
T80477	Muscarinic toxin 3 (MT3) 是高效的非竞争性mAChR及adrenoceptors拮抗剂，对M1、M4、α1A、α1B、α1D、α2A、α2B、α2C受体展示出不同程度的选择性，其pIC50值分别为6.71、8.79、8.86、7.57、8.13、8.49、6.5、7.29。该化合物具有显著的肾上腺...
TN1797	Isorhoifolin 异野漆树苷	552-57-8	98%
TN1797	Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
T81798	Mibenratide TFA 化合物 Mibenratide TFA		98%
T81798	Mibenratide TFA，一种小环肽及肾上腺素能 β1 受体 (adrenergic β1 receptor) 拮抗剂，适用于心力衰竭研究。
T15042	D2343 化合物 T15042	72734-63-5	98%
T15042	D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
T6663	Scopine hydrochloride 盐酸东莨菪醇	85700-55-6	98%
T6663	Scopine hydrochloride (6,7-Epoxytropine hydrochloride) 是一种 Anisodine 的代谢物。
T16769	Ro 363 化合物 T16769	74513-77-2	98%
T16769	RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
TN2267	Tetrahydroalstonine 四氢鸭脚木碱	6474-90-4	98%
TN2267	Tetrahydroalstonine 是从 Rhazya stricta 的果实中提取出来的吲哚类生物碱，是一种具有选择性的 α2-肾上腺素受体拮抗剂。Tetrahydroalstonine 在Rauwolfia tetraphylla 中表现出抗精神病活性。
TN3368	Akuammigine 化合物 TN3368	642-17-1	98%
TN3368	Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T11786	KUL-7211 racemate 化合物 T11786	911196-40-2	98%
T11786	KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
T12815	(S)-Terazosin (S)-特拉唑嗪	109351-33-9	98%
T12815	(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T13285	Vatinoxan hydrochloride 化合物 T13285	130466-38-5	98%
T13285	Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
T11036	Diacetolol D7 化合物 T11036	1346604-19-0	98%
T11036	Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.