Sirtuin inhibitor/activator kit 包含Sirtuin 抑制剂/激活剂,Sirtuin 是一种高度保守的去乙酰化酶类蛋白家族,调控蛋白质的翻译后修饰,影响蛋白质的催化活性、稳定性以及与其它蛋白质或染色质结合的能力。Sirtuin 在细胞凋亡、细胞应激反应、衰老、胰岛素分泌、线粒体生物合成、脂质代谢和脂肪酸氧化等方面起着重要作用。TargetMol 为您提供32种精选Sirtuin 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1887 | Inauhzin | 309271-94-1 | 469.58 | 10mM | MDM-2/p53; Sirtuin |
T1919 | Tenovin-1 | 380315-80-0 | 369.48 | 10mM | Autophagy; Dehydrogenase; MDM-2/p53; Mdm2; p53; Sirtuin |
T2412 | SRT1720 hydrochloride | 1001645-58-4 | 506.22 | 10mM | Sirtuin |
T3447 | Thiomyristoyl | 1429749-41-6 | 581.85 | 10mM | Sirtuin |
T3953 | Salermide | 1105698-15-4 | 394.47 | 10mM | Apoptosis; Sirtuin |
T4062 | CAY10602 | 374922-43-7 | 418.44 | 10mM | Sirtuin |
T4108 | 3-TYP | 120241-79-4 | 146.15 | 10mM | Sirtuin |
T4328 | OSS_128167 | 887686-02-4 | 366.33 | 10mM | HBV; Sirtuin |
T6111 | Selisistat | 49843-98-3 | 248.71 | 10mM | Sirtuin |
T6371 | AGK2 | 304896-28-4 | 434.27 | 10mM | Apoptosis; Sirtuin |
T6984 | SirReal2 | 709002-46-0 | 420.55 | 10mM | Sirtuin |
T5490 | AK-7 | 420831-40-9 | 437.35 | 10mM | Sirtuin |
T5618 | AK-1 | 330461-64-8 | 403.45 | 10mM | Sirtuin |
T8346 | SRT 1460 | 925432-73-1 | 507.6 | 10mM | Sirtuin |
T16932 | SRT 2183 | 1001908-89-9 | 468.57 | 10mM | Apoptosis; Sirtuin |
T8480 | Tenovin-6 Hydrochloride | 1011301-29-3 | 491.09 | 10mM | Autophagy; Dehydrogenase; HDAC; MDM-2/p53; p53; Sirtuin |
T21679 | 4'-bromo-Resveratrol | 1224713-90-9 | 291.14 | 10mM | Sirtuin |
T9106 | E1231 | 1031195-19-3 | 363.41 | 10mM | Sirtuin |
T12919 | SIRT-IN-2 | 1431411-66-3 | 383.49 | 10mM | Sirtuin |
T9320 | YK-3-237 | 1215281-19-8 | 372.18 | 10mM | Sirtuin |
T50080 | MC2184 | 74901-20-5 | 214.18 | 10mM | Sirtuin |
TN7093 | N-Caffeoyltryptophan | 109163-69-1 | 366.37 | 10mM | Sirtuin |
T7058 | Selisistat S-enantiomer | 848193-68-0 | 248.71 | 10mM | Sirtuin |
T39233 | SIRT7 inhibitor 97491 | 1807758-81-1 | 285.73 | 10mM | Sirtuin |
T12918 | SIRT-IN-1 | 1431411-60-7 | 389.52 | 10mM | Sirtuin |
T9998 | 4H-1,2,4-Triazole, 3-(phenoxymethyl)-4-phenyl-5-[(phenylmethyl)thio]- | 129544-85-0 | 373.47 | 10mM | Sirtuin |
T9648 | SIRT1-IN-1 | 352554-02-0 | 228.29 | 10mM | Sirtuin;Antiviral |
T12922 | Sirtuin modulator 1 | 2070015-26-6 | 606.2 | 10mM | Sirtuin |
T35347 | Et-29 | 2166487-23-4 | 666.83 | 10mM | Sirtuin |
T22094 | JGB1741 | 1256375-38-8 | 440.56 | 10mM | Sirtuin |
T28543 | RK-9123016 | 955900-27-3 | 374.42 | 10mM | Sirtuin |
T12920 | Sirt2-IN-1 | 1862238-00-3 | 557.69 | 10mM | Sirtuin |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |