PKC inhibitor kit 包含蛋白激酶C PKC 抑制剂,在第二信使存在时,PKC 成为膜结合的酶,作用于细胞质中的酶和细胞核中的转录因子, 参与糖代谢、细胞分化、基因表达的调控与长时程抑制,如受体脱敏、调节膜结构、调节转录、介导免疫应答、调节细胞生长以及学习和记忆等。TargetMol 为您提供40种精选PKC 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
TN1299 | Desmethylglycitein | 17817-31-1 | 270.2 | 10mM | CDK; PI3K; PKC |
T14072 | A-443654 | 552325-16-3 | 397.47 | 10mM | Akt; Casein Kinase; CDK; Chk; ERK; FLT; GSK-3; MAPK; PKA; PKC; S6 Kinase; Src; VEGFR |
T4444 | A-674563 HCl (552325-73-2(free base)) | T4444 | 394.9 | 10mM | Akt; CDK; ERK; PKA; PKC |
T7659 | Bisindolylmaleimide IV | 119139-23-0 | 327.34 | 10mM | PKC |
T10549 | Bisindolylmaleimide VIII acetate | 138516-31-1 | 458.51 | 10mM | Apoptosis; PKC |
T6S0052 | Chelerythrine | 34316-15-9 | 348.37 | 10mM | Apoptosis; Autophagy; Bcl; PKC |
T3684 | CP21R7 | 125314-13-8 | 317.3 | 10mM | GSK-3; PKC |
T0979 | Dequalinium chloride | 522-51-0 | 527.59 | 10mM | PKC; Potassium Channel |
T6280 | Enzastaurin | 170364-57-5 | 515.61 | 10mM | Apoptosis; Autophagy; PKC |
T3060 | Fasudil hydrochloride | 105628-07-7 | 327.83 | 10mM | Autophagy; Calcium Channel; HIV Protease; PKA; PKC; ROCK; Serine/threonin kinase |
T6513 | Bisindolylmaleimide I | 133052-90-1 | 412.48 | 10mM | PDGFR; PKC |
T6313 | Go 6983 | 133053-19-7 | 442.51 | 10mM | PKC |
T6285 | GSK-690693 | 937174-76-0 | 425.48 | 10mM | Akt; AMPK; Autophagy; PKC; Serine Protease |
T27525 | HA-1004 | 91742-10-8 | 293.35 | 10mM | PKA;PKC;Serine/threonin kinase |
T5771 | Hypocrellin A | 77029-83-5 | 546.52 | 10mM | Antibacterial; Parasite; PKC |
T5600 | Darovasertib | 1874276-76-2 | 472.47 | 10mM | PKC |
T0033 | Miltefosine | 58066-85-6 | 407.58 | 10mM | Akt; HIV Protease; PKC |
T0158 | Mitoxantrone dihydrochloride | 70476-82-3 | 517.4 | 10mM | PKC; Topoisomerase |
T9256 | N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine | 1071135-06-2 | 388.51 | 10mM | PKC; Serine/threonin kinase |
T0610 | Piceatannol | 10083-24-6 | 244.24 | 10mM | Apoptosis; Autophagy; PKA; PKC; Serine/threonin kinase; Syk |
T3211 | Midostaurin | 120685-11-2 | 570.64 | 10mM | PKC |
T8764 | PKC-iota inhibitor 1 | 2328094-11-5 | 374.4 | 10mM | PKC |
T9863 | PKCiota-IN-2 | 2230055-52-2 | 395.46 | 10mM | PKC |
T5817 | PKC-theta inhibitor | 2253640-49-0 | 454.4 | 10mM | PKC |
T8376 | PKCβ inhibitor 1 | 257879-35-9 | 411.5 | 10mM | Apoptosis; PKC |
T35827L | PKCε Inhibitor Peptide acetate | T35827L | 904.02 | 10mM | PKC |
T5796 | Plantainoside D | 147331-98-4 | 640.6 | 10mM | PKC; RAAS |
T60109 | Protein kinase inhibitor H-7 | 84477-87-2 | 291.37 | 10mM | PKC |
T6643 | Ro 31-8220 Mesylate | 138489-18-6 | 553.65 | 10mM | PKC |
T2356 | Ro-3306 | 872573-93-8 | 351.45 | 10mM | Apoptosis; CDK; ERK; PKA; PKC; SGK |
T16791 | Rottlerin | 82-08-6 | 516.54 | 10mM | Apoptosis; Autophagy; CaMK; HIV Protease; PKA; PKC |
T9605 | Sangivamycin | 18417-89-5 | 309.28 | 10mM | PKC;Nucleoside Antimetabolite/Analog |
T6278 | Sotrastaurin | 425637-18-9 | 438.48 | 10mM | PKC |
T6680 | Staurosporine | 62996-74-1 | 466.53 | 10mM | Antibacterial; Antibiotic; Antifungal; Apoptosis; PKA; PKC; Src |
T4391 | Syk Inhibitor II (hydrochloride) | 227449-73-2 | 413.22 | 10mM | BTK; PKC; Syk; Tyrosine Kinases |
T2441 | TAS-301 | 193620-69-8 | 357.4 | 10mM | PKC |
T17148 | TPPB | 497259-23-1 | 501.54 | 10mM | PKC |
T7604 | Valrubicin | 56124-62-0 | 723.64 | 10mM | Antibiotic; PKC |
T13384L | Y-33075 dihydrochloride | 173897-44-4 | 353.25 | 10mM | CaMK; PKC; ROCK |
T35407 | Ζ-Stat | 3316-02-7 | 384.36 | 10mM | PKC |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |