PKA/cAMP inhibitor/activator kit 包含 PKA/cAMP 抑制剂/激活剂,G 蛋白偶联受体首先将信号传至腺苷酸环化酶,调节 cAMP 的含量,cAMP 决定PKA 的活性,PKA 负责很多蛋白的磷酸化,比如受体、离子通道、转录因子等,这是细胞快速应答胞外信号的过程。还有一类细胞缓慢应答胞外信号的过程,是cAMP 信号通路对细胞基因表达的影响。TargetMol 为您提供34种精选PKA/cAMP 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0465 | Ellagic acid | 476-66-4 | 302.19 | 10mM | Carbonic Anhydrase; Casein Kinase; Endogenous Metabolite; Hedgehog/Smoothened; PKA; PKC; Reactive Oxygen Species; Syk; Topoisomerase |
T0610 | Piceatannol | 10083-24-6 | 244.24 | 10mM | Apoptosis; Autophagy; PKA; PKC; Serine/threonin kinase; Syk |
T0830 | Bithionol | 97-18-7 | 356.04 | 10mM | cAMP; Parasite |
T1418 | Bucladesine sodium | 16980-89-5 | 491.37 | 10mM | PDE; PKA |
T1920 | Capivasertib | 1143532-39-1 | 428.92 | 10mM | Akt; Autophagy; mTOR; PKA |
T2205 | Acefylline | 652-37-9 | 238.2 | 10mM | Adenosine Receptor; HDAC; PAD; PDE; PKA; TNF |
T2244 | ESI-09 | 263707-16-0 | 330.77 | 10mM | cAMP; Virus Protease |
T2356 | Ro-3306 | 872573-93-8 | 351.45 | 10mM | Apoptosis; CDK; ERK; PKA; PKC; SGK |
T2482 | AT13148 | 1056901-62-2 | 313.78 | 10mM | Akt; PKA; ROCK; S6 Kinase; SGK |
T2851 | Daphnetin | 486-35-1 | 178.14 | 10mM | Autophagy; EGFR; Parasite; PKA; PKC |
T3050 | ML-7 hydrochloride | 110448-33-4 | 452.74 | 10mM | Myosin; PKA; PKC; Serine/threonin kinase; YAP |
T3060 | Fasudil hydrochloride | 105628-07-7 | 327.83 | 10mM | Autophagy; Calcium Channel; HIV Protease; PKA; PKC; ROCK; Serine/threonin kinase |
T3269 | Metadoxine | 74536-44-0 | 298.29 | 10mM | 5-HT Receptor; PKA |
T4444 | A-674563 HCl (552325-73-2(free base)) | T4444 | 394.9 | 10mM | Akt; CDK; ERK; PKA; PKC |
T6250 | H-89 dihydrochloride | 130964-39-5 | 519.28 | 10mM | Autophagy; PKA; S6 Kinase |
T6304 | AT7867 | 857531-00-1 | 337.85 | 10mM | Akt; PKA; S6 Kinase |
T6536 | HJC0350 | 885434-70-8 | 277.38 | 10mM | cAMP |
T6680 | Staurosporine | 62996-74-1 | 466.53 | 10mM | Antibacterial; Antibiotic; Antifungal; Apoptosis; PKA; PKC; Src |
T6747 | 8-Bromo-cAMP sodium salt | 76939-46-3 | 430.08 | 10mM | PKA |
T4S2128 | Bilobetin | 521-32-4 | 552.49 | 10mM | PKA; PPAR |
T7648 | HA-100 | 84468-24-6 | 277.34 | 10mM | Myosin; PKA; PKC |
T15485 | HJC0197 | 1383539-73-8 | 339.45 | 10mM | cAMP; Ras |
T14069 | A-3 hydrochloride | 78957-85-4 | 321.22 | 10mM | CaMK; Casein Kinase; PKA; PKC |
TN1334 | 7-Methoxyrosmanol | 113085-62-4 | 360.45 | 10mM | cAMP |
T6139L | A-674563 2HCl(552325-73-2(fb-2hcl)) | T6139L | 431.36 | 10mM | Akt; CDK; ERK; PKA; PKC |
T15247 | ESI-05 | 5184-64-5 | 274.38 | 10mM | cAMP |
TP1789L | Malantide acetate(86555-35-3 free base) | TP1789L | 1693.97 | 10mM | PKA; PKC |
T12616L | CE3F4 | 143703-25-7 | 351.01 | 10mM | cAMP |
T15658 | KH7 | 330676-02-3 | 419.3 | 10mM | AChR; cAMP |
T21983L | PKI 14-22 amide, myristoylated Acetate | T21983L | 1269.54 | 10mM | PKA |
T21674L | PKA inhibitor fragment (6-22) amide Acetate | T21674L | 1928.11 | 10mM | PKA |
T9613 | TDI-10229 | T9613 | 313.79 | 10mM | cAMP |
T27525 | HA-1004 | 91742-10-8 | 293.35 | 10mM | PKA;PKC;Serine/threonin kinase |
T11212 | EPAC 5376753 | 302826-61-5 | 367.21 | 10mM | cAMP |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |