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PKA/cAMP inhibitor/activator kit

PKA/cAMP inhibitor/activator kit

产品编号 CL0143 PKA/cAMP inhibitor/activator kit
  库化合物信息   Excel SDF

PKA/cAMP inhibitor/activator kit 包含 PKA/cAMP 抑制剂/激活剂,G 蛋白偶联受体首先将信号传至腺苷酸环化酶,调节 cAMP 的含量,cAMP 决定PKA 的活性,PKA 负责很多蛋白的磷酸化,比如受体、离子通道、转录因子等,这是细胞快速应答胞外信号的过程。还有一类细胞缓慢应答胞外信号的过程,是cAMP 信号通路对细胞基因表达的影响。TargetMol 为您提供34种精选PKA/cAMP 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
10 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品组成

IDCompoundCASMWConcentrationTarget
T0465Ellagic acid476-66-4302.1910mMCarbonic Anhydrase; Casein Kinase; Endogenous Metabolite; Hedgehog/Smoothened; PKA; PKC; Reactive Oxygen Species; Syk; Topoisomerase
T0610Piceatannol10083-24-6244.2410mMApoptosis; Autophagy; PKA; PKC; Serine/threonin kinase; Syk
T0830Bithionol97-18-7356.0410mMcAMP; Parasite
T1418Bucladesine sodium16980-89-5491.3710mMPDE; PKA
T1920Capivasertib1143532-39-1428.9210mMAkt; Autophagy; mTOR; PKA
T2205Acefylline652-37-9238.210mMAdenosine Receptor; HDAC; PAD; PDE; PKA; TNF
T2244ESI-09263707-16-0330.7710mMcAMP; Virus Protease
T2356Ro-3306872573-93-8351.4510mMApoptosis; CDK; ERK; PKA; PKC; SGK
T2482AT131481056901-62-2313.7810mMAkt; PKA; ROCK; S6 Kinase; SGK
T2851Daphnetin486-35-1178.1410mMAutophagy; EGFR; Parasite; PKA; PKC
T3050ML-7 hydrochloride110448-33-4452.7410mMMyosin; PKA; PKC; Serine/threonin kinase; YAP
T3060Fasudil hydrochloride105628-07-7327.8310mMAutophagy; Calcium Channel; HIV Protease; PKA; PKC; ROCK; Serine/threonin kinase
T3269Metadoxine74536-44-0298.2910mM5-HT Receptor; PKA
T4444A-674563 HCl (552325-73-2(free base))T4444394.910mMAkt; CDK; ERK; PKA; PKC
T6250H-89 dihydrochloride130964-39-5519.2810mMAutophagy; PKA; S6 Kinase
T6304AT7867857531-00-1337.8510mMAkt; PKA; S6 Kinase
T6536HJC0350885434-70-8277.3810mMcAMP
T6680Staurosporine62996-74-1466.5310mMAntibacterial; Antibiotic; Antifungal; Apoptosis; PKA; PKC; Src
T67478-Bromo-cAMP sodium salt76939-46-3430.0810mMPKA
T4S2128Bilobetin521-32-4552.4910mMPKA; PPAR
T7648HA-10084468-24-6277.3410mMMyosin; PKA; PKC
T15485HJC01971383539-73-8339.4510mMcAMP; Ras
T14069A-3 hydrochloride78957-85-4321.2210mMCaMK; Casein Kinase; PKA; PKC
TN13347-Methoxyrosmanol113085-62-4360.4510mMcAMP
T6139LA-674563 2HCl(552325-73-2(fb-2hcl))T6139L431.3610mMAkt; CDK; ERK; PKA; PKC
T15247ESI-055184-64-5274.3810mMcAMP
TP1789LMalantide acetate(86555-35-3 free base)TP1789L1693.9710mMPKA; PKC
T12616LCE3F4143703-25-7351.0110mMcAMP
T15658KH7330676-02-3419.310mMAChR; cAMP
T21983LPKI 14-22 amide, myristoylated AcetateT21983L1269.5410mMPKA
T21674LPKA inhibitor fragment (6-22) amide AcetateT21674L1928.1110mMPKA
T9613TDI-10229T9613313.7910mMcAMP
T27525HA-100491742-10-8293.3510mMPKA;PKC;Serine/threonin kinase
T11212EPAC 5376753302826-61-5367.2110mMcAMP

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

产品优势

  • 靶点明确
  • 产品精选
  • 试剂新鲜

产品应用

  • 信号通路研究
  • 预实验探索

包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (CL0143)
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化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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