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PDGFR inhibitor kit

PDGFR inhibitor kit

产品编号 CL0071 PDGFR inhibitor kit
  库化合物信息   Excel SDF

PDGFR inhibitor kit 包含血小板衍生生长因子受体 PDGFR 抑制剂,PDGF 受体能够促进细胞的趋化、分裂与增殖、机体生长发育、创伤修复,在调控细胞增殖、分化、生长、发育上扮演相当重要的角色,PDGF 及其受体的高表达促进肿瘤生成,PDGFR 基因突变也可导致肿瘤。PDGFR 抑制剂使肿瘤细胞失去能量来源导致细胞凋亡。TargetMol 为您提供48种精选 PDGFR 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
10 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品组成

IDCompoundCASMWConcentrationTarget
T0093LSorafenib284461-73-0464.8310mMApoptosis; Autophagy; c-Kit; Ferroptosis; FLT; PDGFR; Raf; VEGFR
T0097LPazopanib444731-52-6437.5210mMAutophagy; c-Kit; FGFR; PDGFR; VEGFR
T0374LSunitinib557795-19-4398.4710mMApoptosis; Autophagy; c-Kit; FLT; IRE1; Mitophagy; PDGFR; VEGFR
T1452Axitinib319460-85-0386.4710mMc-Kit; PDGFR; VEGFR
T1667Tandutinib387867-13-2562.710mMApoptosis; c-Kit; CSF-1R; FLT; PDGFR; Src
T1777Nintedanib656247-17-5539.6210mMFGFR; FLT; PDGFR; Src; VEGFR
T1792Regorafenib755037-03-7482.8210mMAutophagy; c-Kit; c-RET; PDGFR; Raf; VEGFR
T1836AZD2932883986-34-3447.4910mMc-Kit; FLT; PDGFR; VEGFR
T2070Agerafenib1188910-76-0517.4610mMBcr-Abl; c-Kit; c-RET; PDGFR; Raf; Src
T2358ENMD-2076934353-76-1375.4710mMApoptosis; Aurora Kinase; c-RET; FGFR; FLT; PDGFR; Src; VEGFR
T2372Ponatinib943319-70-8532.5610mMAutophagy; Bcr-Abl; c-Kit; FGFR; PDGFR; Src; VEGFR
T2415PP1211092788-83-4319.3610mMApoptosis; Bcr-Abl; Hck; mTOR; PDGFR; Src; VEGFR
T2456Tivozanib475108-18-0454.8610mMEphrin Receptor; PDGFR; VEGFR
T2479Tyrphostin A910537-47-0282.3810mMEGFR; Influenza Virus; PDGFR; VEGFR
T2500Cediranib288383-20-0450.5110mMAutophagy; c-Kit; FLT; PDGFR; VEGFR
T2514Linifanib796967-16-3375.410mMApoptosis; Autophagy; c-Fms; c-Kit; CSF-1R; FLT; PDGFR; VEGFR
T2516Amuvatinib850879-09-3447.5110mMApoptosis; c-Kit; c-Met/HGFR; c-RET; DNA/RNA Synthesis; FLT; PDGFR
T2609Masitinib790299-79-5498.6410mMApoptosis; Bcr-Abl; c-Fms; c-Kit; FAK; FGFR; Hck; PDGFR; Src
T2677Crenolanib670220-88-9443.5410mMAutophagy; FLT; PDGFR
T3463NVP-ACC789300842-64-2405.310mMPDGFR; VEGFR
T3476JI-101900573-88-8466.3410mMEphrin Receptor; PDGFR; VEGFR
T6091CP-673451343787-29-1417.510mMc-Kit; PDGFR; VEGFR
T6166Telatinib332012-40-5409.8310mMc-Kit; PDGFR; VEGFR
T6184Orantinib252916-29-3310.3510mMApoptosis; FGFR; PDGFR; VEGFR
T6230Imatinib152459-95-5493.610mMAutophagy; Bcr-Abl; c-Kit; PDGFR; SARS-CoV
T6479Dovitinib lactate hydrate915769-50-5482.5110mMc-Kit; FGFR; FLT; PDGFR; VEGFR
T6711Tyrphostin AG1296146535-11-7266.2910mMApoptosis; c-Kit; FGFR; FLT; PDGFR
T6920ON1233001357470-29-1429.5210mMAMPK; c-RET; CDK; FGFR; JAK; PDGFR; Src
T5001Nintedanib esylate656247-18-6649.7610mMFGFR; PDGFR; VEGFR
T5109Avapritinib1703793-34-3498.5610mMc-Kit; PDGFR; PDGFR
T5466Tyrosine kinase-IN-1705946-27-6445.5410mMFGFR; FLT; PDGFR; VEGFR
T7394Toceranib Phosphate874819-74-6494.4510mMc-Kit; PDGFR; Tyrosinase; VEGFR
T7945SU14813627908-92-3442.4810mMc-Kit; PDGFR; VEGFR
T8491Vorolanib1013920-15-4439.4810mMPDGFR; VEGFR
T8482Ripretinib1442472-39-0510.3610mMApoptosis; c-Kit; FLT; PDGFR; VEGFR
T8541Lenvatinib mesylate857890-39-2522.9610mMc-Kit; c-RET; FGFR; PDGFR; VEGFR
T10157Regorafénib N-oxyde (M2)835621-11-9498.8110mMc-Kit; c-RET; Drug Metabolite; PDGFR; Raf; VEGFR
T15616JNJ-10198409627518-40-5325.3410mMPDGFR
T16750Rigosertib592542-59-1451.4910mMApoptosis; Bcr-Abl; CDK; FLT; PDGFR; PI3K; PLK; Src
T12145LN-Desethylsunitinib hydrochloride1261432-05-6406.8810mMc-Kit; PDGFR; VEGFR
T8900Seralutinib1619931-27-9469.5510mMPDGFR
TQ0235AC7101351522-04-7562.710mMc-Kit; FLT; PDGFR
T16975TAK-5931005780-62-0445.4710mMPDGFR; VEGFR
T13238Tyrphostin AG1433168835-90-3266.2910mMPDGFR; VEGFR
T35570Chiauranib1256349-48-0435.4710mMVEGFR;PDGFR;c-Kit;Aurora Kinase;c-Fms;FLT
T41003KG5877874-85-6459.4510mMRaf;PDGFR;FLT;c-Kit
T16947SU16f251356-45-3386.4410mMPDGFR
T13824PP58212391-58-7456.3310mMPDGFR;FGFR;Src;p38 MAPK;TNF

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

产品优势

  • 靶点明确
  • 产品精选
  • 试剂新鲜

产品应用

  • 信号通路研究
  • 预实验探索

包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (CL0071)
点击图片重新获取验证码

化合物库组成

PDGFR (48)
VEGFR (32)
c-Kit (28)
FLT (18)
FGFR (13)
Apoptosis (12)
Src (10)
Autophagy (9)
c-RET (7)
Bcr-Abl (6)
Raf (5)
c-Fms (3)
CDK (2)
CSF-1R (2)
Ephrin Receptor (2)
Aurora Kinase (2)
Hck (2)
JAK (1)
mTOR (1)
p38 MAPK (1)
FAK (1)
SARS-CoV (1)
Drug Metabolite (1)
DNA/RNA Synthesis (1)
Tyrosinase (1)
c-Met/HGFR (1)
PI3K (1)
AMPK (1)
PLK (1)
IRE1 (1)
Ferroptosis (1)
EGFR (1)
Mitophagy (1)
TNF (1)
Influenza Virus (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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