PARP inhibitor kit 包含多聚 ADP 核糖聚合酶 PARP 抑制剂,PARP 催化 ADP 核糖残基从 NAD+转移到目标底物上,构建一个多聚 ADP 核糖,可以指导DNA 修复、维持基因组完整性,并调控多种代谢和信号转导过程等。PARP 抑制剂能够影响癌细胞的自我复制方式,可以用于卵巢癌、前列腺癌以及胰腺癌等遗传性癌症的治疗研究。TargetMol 为您提供41种精选PARP 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T2105 | Veliparib dihydrochloride | 912445-05-7 | 317.21 | 10mM | Autophagy; PARP |
T2484 | AZD-2461 | 1174043-16-3 | 395.43 | 10mM | PARP |
T3015 | Olaparib | 763113-22-0 | 434.46 | 10mM | Autophagy; Mitophagy; PARP |
T6181 | UPF 1069 | 1048371-03-4 | 279.29 | 10mM | PARP |
T6197 | PJ34 | 344458-19-1 | 295.34 | 10mM | PARP |
T6224 | Iniparib | 160003-66-7 | 292.03 | 10mM | Influenza Virus; PARP |
T6253 | Talazoparib | 1207456-01-6 | 380.35 | 10mM | PARP |
T6329 | 3-Aminobenzamide | 3544-24-9 | 136.15 | 10mM | PARP |
T6339 | AG14361 | 328543-09-5 | 320.39 | 10mM | PARP |
T6366 | A-966492 | 934162-61-5 | 324.35 | 10mM | PARP |
T6578 | ME0328 | 1445251-22-8 | 321.37 | 10mM | PARP |
T6780 | Benzamide | 55-21-0 | 121.14 | 10mM | Endogenous Metabolite; PARP |
T6912 | NU1025 | 90417-38-2 | 176.17 | 10mM | PARP |
T7042 | 1,5-Isoquinolinediol | 5154-02-9 | 161.16 | 10mM | PARP |
T5399 | GeA-69 | 2143475-98-1 | 300.36 | 10mM | PARP |
T7439 | 3-Methoxybenzamide | 5813-86-5 | 151.16 | 10mM | Antibacterial; PARP; Transferase |
T7896 | BYK204165 | 1104546-89-5 | 252 | 10mM | PARP |
T8150 | Nudifloramide | 701-44-0 | 152.15 | 10mM | Endogenous Metabolite; PARP |
T21524 | 4-amino-1,8-Naphthalimide | 1742-95-6 | 212.2 | 10mM | PARP |
T22414 | RBN012759 | 2360851-29-0 | 378.46 | 10mM | PARP |
T12695 | RBN-2397 | 2381037-82-5 | 523.43 | 10mM | PARP |
T16807 | Rucaparib monocamsylate | 1859053-21-6 | 555.66 | 10mM | PARP |
T8806 | Fluzoparib | 1358715-18-0 | 472.4 | 10mM | PARP |
T22264 | AZ9482 | 1825345-33-2 | 450.5 | 10mM | PARP |
T4471 | E7449 | 1140964-99-3 | 317.3 | 10mM | PARP |
T5058 | Pamiparib | 1446261-44-4 | 298.31 | 10mM | PARP |
T9024 | OUL35 | 6336-34-1 | 256.26 | 10mM | PARP |
T4472 | NMS-P118 | 1262417-51-5 | 395.42 | 10mM | PARP |
T22749 | DR2313 | 284028-90-6 | 182.24 | 10mM | PARP |
T9165 | AZD5305 | 2589531-76-8 | 406.48 | 10mM | PARP |
T12064 | Niraparib (R-enantiomer) | 1038915-58-0 | 320.39 | 10mM | PARP |
T50098 | TIQ-A | 420849-22-5 | 201.24 | 10mM | PARP |
T50044 | 5-amino-1,2-dihydroisoquinolin-1-one | 93117-08-9 | 160.17 | 10mM | PARP |
T9497 | Niraparib tosylate monohyrate | 1613220-15-7 | 492.59 | 10mM | PARP |
T9430 | Venadaparib | 1681017-83-3 | 406.45 | 10mM | PARP |
T22988 | MK-4827 Racemate | 1038915-75-1 | 320.39 | 10mM | PARP |
T9593 | Senaparib | 1401682-78-7 | 478.45 | 10mM | PARP |
T9610 | PARP1-IN-5 dihydrochloride | T9610 | 537.46 | 10mM | PARP |
T9891 | PARP1-IN-8 | 836640-15-4 | 403.86 | 10mM | PARP |
T9756 | AZD-9574 | 2756333-39-6 | 428.44 | 10mM | PARP |
T11143 | EB-47 | 366454-36-6 | 537.53 | 10mM | PARP |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |