Notch pathway inhibitor kit 包含 Notch 通路抑制剂,Notch 基因编码高度保守的细胞表面受体,调节多种生物细胞发育的多个过程,包括多能祖细胞的分化、细胞凋亡、细胞增殖及细胞边界的形成。Notch 通路抑制剂可以抑制促生长基因如cyclin D1和C-myc 的表达,抑制PI3K/AKT 等抗凋亡通路。TargetMol 为您提供17种精选Notch 通路抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T2842 | Tangeretin | 481-53-8 | 372.38 | 10mM | Apoptosis; Gamma-secretase |
T3075 | FLI-06 | 313967-18-9 | 438.52 | 10mM | Gamma-secretase |
T3399 | Psoralidin | 18642-23-4 | 336.34 | 10mM | Akt; Antibacterial; COX; Estrogen/progestogen Receptor; Gamma-secretase; Lipoxygenase; Reactive Oxygen Species |
T3540 | IMR-1A | 331862-41-0 | 325.36 | 10mM | Drug Metabolite; Gamma-secretase |
T3633 | Crenigacestat | 1421438-81-4 | 464.44 | 10mM | Gamma-secretase |
T6063 | LY-411575 | 209984-57-6 | 479.48 | 10mM | Apoptosis; Gamma-secretase |
T6125 | Semagacestat | 425386-60-3 | 361.44 | 10mM | Beta Amyloid; Gamma-secretase |
T6135 | YO-01027 | 209984-56-5 | 463.48 | 10mM | Gamma-secretase |
T6202 | DAPT | 208255-80-5 | 432.46 | 10mM | Apoptosis; Autophagy; Beta Amyloid; Gamma-secretase |
T6249 | Avagacestat | 1146699-66-2 | 520.88 | 10mM | Gamma-secretase |
T6274 | RO4929097 | 847925-91-1 | 469.4 | 10mM | Beta Amyloid; Gamma-secretase |
T6861 | IMR-1 | 310456-65-6 | 353.41 | 10mM | Gamma-secretase |
T4S1990 | Carvacrol | 499-75-2 | 150.22 | 10mM | Antifungal; Apoptosis; Endogenous Metabolite; Gamma-secretase |
TWS2045 | Bruceine D | 21499-66-1 | 410.41 | 10mM | Antiviral; Apoptosis; Gamma-secretase; Parasite |
T12246 | CB-103 | 218457-67-1 | 242.32 | 10mM | Gamma-secretase |
T13410 | ZLDI-8 | 667880-38-8 | 433.52 | 10mM | Apoptosis; Gamma-secretase; Immunology/Inflammation related; Phosphatase |
T6935 | Nirogacestat | 1290543-63-3 | 489.64 | 10mM | Apoptosis; Gamma-secretase |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |