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MEK inhibitor kit

MEK inhibitor kit

现 货
产品编号 CL0091 MEK inhibitor kit
  库化合物信息   Excel SDF

MEK inhibitor kit 包含丝裂原活化/细胞外信号调节激酶 MEK 抑制剂,MEK 可磷酸化靶蛋白上 Ser/Thr 和Tyr 残基,是RAS/RAF-MEK-ERK 信号转导通路的主要组分。MEK 信号通路参与了细胞周期进行、细胞凋亡、迁移、分化、代谢和增殖等过程的调节,MEK 表达水平及其结构的改变与癌症等多种疾病的发生密切相关。TargetMol 为您提供34种精选MEK 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
10 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品组成

IDCompoundCASMWConcentrationTarget
T0468Lidocaine137-58-6234.3410mMApoptosis; ERK; Histamine Receptor; MEK; NF-κB; Sodium Channel
T1144Lidocaine hydrochloride73-78-9270.810mMApoptosis; ERK; MEK; NF-κB; Sodium Channel
T2125Trametinib871700-17-3615.3910mMApoptosis; Autophagy; MEK
T2327Pelitinib257933-82-7467.9210mMEGFR; MEK; Raf; Src
T2378RGB-286638 free base784210-88-4545.6310mMCDK; GSK-3; JAK; MEK
T2416BIX021891094614-85-3440.5410mMERK; MEK; TGF-beta/Smad
T2443CI-1040212631-79-3478.6710mMApoptosis; MEK
T2508Binimetinib606143-89-9441.2310mMAutophagy; MEK
T2623PD98059167869-21-8267.2810mMAryl Hydrocarbon Receptor; Autophagy; ERK; MEK
T2708SL327305350-87-2335.3510mMDNA/RNA Synthesis; MEK
T2836Isorhamnetin480-19-3316.2710mMEndogenous Metabolite; MEK; PI3K
T3623Cobimetinib934660-93-2531.3210mMApoptosis; MEK
T6083AZD8330869357-68-6461.2310mMERK; MEK
T6131Pimasertib1236699-92-5431.210mMMEK
T6152PD318088391210-00-7561.0910mMMEK
T6189Mirdametinib391210-10-9482.1910mMApoptosis; Autophagy; MEK
T6218Selumetinib606143-52-6457.6810mMApoptosis; ERK; MEK
T6324BIX021881094614-84-2412.4810mMERK; MEK; TGF-beta/Smad
T6419BMS-536924468740-43-4479.9610mMApoptosis; FAK; IGF-1R; MEK; Src
T6692TAK-7331035555-63-5504.2310mMMEK
T6760APS-2-79 hydrochloride2002381-31-7423.8910mMMAPK; MEK
T6785BI-8473251207293-36-4464.5610mMApoptosis; Aurora Kinase; MEK
T6971Ro 5126766946128-88-7471.4610mMMEK; Raf
T5S2361Epiberberine6873-09-2336.3610mMAChE; AChR; BACE; Beta-secretase; ERK; MEK
TMS2181trans-Zeatin1637-39-4219.2410mMEndogenous Metabolite; ERK; MEK
T5412RO4987655874101-00-5565.2810mMMEK
T5857Trametinib (DMSO solvate)1187431-43-1693.5310mMApoptosis; MEK
T7742GW 284543 hydrochloride179246-08-3408.8710mMMEK
T21295BIX021891265916-41-3440.5410mMERK; MEK
T9321zapnometinib303175-44-2409.5510mMAntibacterial; Influenza Virus; MEK
T21635PD184161212631-67-9557.5610mMMEK
T27242EF24342808-40-6311.3310mMCaspase; ERK; MEK
T36631BAY-60352247890-13-5396.4810mMHistone Methyltransferase;MEK
T21980PD 198306212631-61-3476.2310mMMEK

化合物库定制

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产品优势

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产品应用

  • 信号通路研究
  • 预实验探索

包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (CL0091)
点击图片重新获取验证码

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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