LPL Receptor antagonist/agonist kit 包含脂蛋白脂肪酶LPL 拮抗剂/激动剂,LPL 是脂肪细胞、心肌细胞、骨骼肌细胞、乳腺细胞以及巨噬细胞等实质细胞合成和分泌的一种糖蛋白,催化脂蛋白中TG 水解,以供组织氧化供能和贮存,参与VLDL 和HDL 之间的载脂蛋白和磷脂的转换。另外,LPL 还具有增加CM 残粒结合到LPL 受体上的能力,促进CM 残粒摄取。TargetMol 为您提供22种精选LPL 拮抗剂/激动剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T2171 | SEW​2871 | 256414-75-2 | 440.36 | 10mM | LPL Receptor; S1P Receptor |
T2539 | Fingolimod hydrochloride | 162359-56-0 | 343.93 | 10mM | LPL Receptor; PAK; S1P Receptor; TRP/TRPV Channel |
T3258 | Ponesimod | 854107-55-4 | 460.97 | 10mM | LPL Receptor; S1P Receptor |
T3961 | CYM-5541 | 945128-26-7 | 316.44 | 10mM | LPL Receptor; S1P Receptor |
T4031 | S1p receptor agonist 1 | 1514888-56-2 | 409.45 | 10mM | LPL Receptor; S1P Receptor |
T6403 | Siponimod | 1230487-00-9 | 516.6 | 10mM | LPL Receptor; S1P Receptor |
T6923 | Ozanimod | 1306760-87-1 | 404.46 | 10mM | LPL Receptor; S1P Receptor |
T7360 | GSK2018682 | 1034688-30-6 | 440.88 | 10mM | LPL Receptor; S1P Receptor |
T7832 | Ibrolipim | 133208-93-2 | 451.25 | 10mM | LPL Receptor |
T7939 | Fingolimod | 162359-55-9 | 307.47 | 10mM | LPL Receptor; PAK; S1P Receptor |
T10305 | Amiselimod hydrochloride | 942398-84-7 | 413.9 | 10mM | LPL Receptor; S1P Receptor |
T17183 | TY-52156 | 934369-14-9 | 364.27 | 10mM | LPL Receptor; S1P Receptor |
T15629 | JTE-013 | 383150-41-2 | 408.29 | 10mM | Apoptosis; LPL Receptor; S1P Receptor |
T8840 | PF-543 hydrochloride | 1706522-79-3 | 502.1 | 10mM | Apoptosis; Autophagy; LPL Receptor; S1P Receptor |
T15032 | CYM50308 | 1345858-76-5 | 405.46 | 10mM | LPL Receptor; S1P Receptor |
T22703 | CYM-5520 | 1449747-00-5 | 345.4 | 10mM | LPL Receptor; S1P Receptor |
TQ0227 | Etrasimod | 1206123-37-6 | 457.48 | 10mM | LPL Receptor; S1P Receptor |
T9199 | GLPG2938 | 2130996-00-6 | 503.4 | 10mM | LPL Receptor; S1P Receptor |
T9464 | CYM50358 | 1314212-39-9 | 389.27 | 10mM | LPL Receptor |
T28169 | NIBR-0213 | 1233332-14-3 | 464.98 | 10mM | LPL Receptor |
T12086 | Mocravimod hydrochloride | 509088-69-1 | 480.45 | 10mM | LPL Receptor |
T12821 | S1PR1 modulator 1 | 2328109-05-1 | 408.51 | 10mM | LPL Receptor |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |