JAK inhibitor kit 包含 Janus 激酶 JAK 抑制剂,JAK 抑制剂阻断 JAK/STAT 信号通路,这是一条与细胞因子密切相关的细胞内信号传导通路,参与细胞的增殖、分化、凋亡以及免疫调节等过程,JAK 抑制剂主要用于血液系统疾病、类风湿性关节炎、肿瘤、及银屑病等疾病的治疗研究。TargetMol 为您提供56种精选 JAK 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1849 | Momelotinib | 1056634-68-4 | 414.46 | 10mM | Apoptosis; Autophagy; JAK |
T1929 | Filgotinib | 1206161-97-8 | 425.5 | 10mM | JAK; Tyrosine Kinases |
T1985 | WHI-P154 | 211555-04-3 | 376.2 | 10mM | Apoptosis; EGFR; JAK; Src; VEGFR |
T1995 | Fedratinib | 936091-26-8 | 524.68 | 10mM | Apoptosis; c-RET; FLT; JAK |
T2035 | WHI-P258 | 21561-09-1 | 281.31 | 10mM | EGFR; JAK; JNK |
T2045 | JANEX-1 | 202475-60-3 | 297.31 | 10mM | JAK |
T2156 | WP1066 | 857064-38-1 | 356.22 | 10mM | Apoptosis; JAK; STAT |
T2360 | Baricitinib phosphate | 1187595-84-1 | 469.41 | 10mM | JAK; Tyrosine Kinases |
T2487 | Cerdulatinib | 1198300-79-6 | 445.54 | 10mM | JAK; Syk; Tyrosine Kinases |
T2636 | Decernotinib | 944842-54-0 | 392.38 | 10mM | JAK; Tyrosine Kinases |
T2638 | Gandotinib | 1229236-86-5 | 469.94 | 10mM | FGFR; FLT; JAK; VEGFR |
T3042 | NSC 42834 | 195371-52-9 | 344.45 | 10mM | JAK |
T3043 | Ruxolitinib phosphate | 1092939-17-7 | 404.36 | 10mM | Autophagy; JAK; Mitophagy |
T3065 | TG101209 | 936091-14-4 | 509.67 | 10mM | Apoptosis; Autophagy; c-RET; FLT; JAK |
T3068 | AT9283 | 896466-04-9 | 381.43 | 10mM | Apoptosis; Aurora Kinase; Autophagy; Bcr-Abl; FLT; JAK |
T3069 | AZD-1480 | 935666-88-9 | 348.77 | 10mM | JAK |
T3072 | XL019 | 945755-56-6 | 444.53 | 10mM | Apoptosis; FLT; JAK; PDGFR |
T3076 | GLPG0634 analog | 1206101-20-3 | 410.43 | 10mM | JAK; Tyrosine Kinases |
T3080 | Pyridone 6 | 457081-03-7 | 309.34 | 10mM | JAK; Tyrosine Kinases |
T3620 | Solcitinib | 1206163-45-2 | 389.45 | 10mM | JAK |
T3673 | Mollugin | 55481-88-4 | 284.3 | 10mM | HER; JAK |
T3998 | Itacitinib | 1334298-90-6 | 553.53 | 10mM | JAK |
T4210 | SAR-20347 | 1450881-55-6 | 444.85 | 10mM | JAK; Tyrosine Kinases |
T4227 | SB1317 hydrochloride (1204918-72-8(free base)) | T4227 | 408.92 | 10mM | CDK; FLT; JAK |
T6020 | Pacritinib | 937272-79-2 | 472.58 | 10mM | FLT; JAK; Tyrosine Kinases |
T6294 | NVP-BSK805 2HCl (1092499-93-8(free base)) | T6294 | 563.47 | 10mM | JAK; Tyrosine Kinases |
T6309 | AZ960 | 905586-69-8 | 354.36 | 10mM | Apoptosis; JAK; Parasite; Virus Protease |
T6321 | Tofacitinib | 477600-75-2 | 312.37 | 10mM | Apoptosis; JAK; ROCK; Src |
T6790 | BMS-911543 | 1271022-90-2 | 432.52 | 10mM | Histone Methyltransferase; JAK; Tyrosine Kinases |
T6838 | FLLL32 | 1226895-15-3 | 464.55 | 10mM | Apoptosis; JAK; STAT |
T6914 | Oclacitinib maleate | 1640292-55-2 | 453.51 | 10mM | JAK; Tyrosine Kinases |
T7503 | Upadacitinib | 1310726-60-3 | 380.37 | 10mM | JAK |
T6122 | CEP-33779 | 1257704-57-6 | 462.57 | 10mM | JAK |
T5091 | FM-381 | 2226521-65-7 | 428.49 | 10mM | JAK |
T5382 | Ritlecitinib | 1792180-81-4 | 285.34 | 10mM | JAK |
T5492 | JAK3-IN-6 | 1443235-95-7 | 350.37 | 10mM | JAK |
T14331 | Gusacitinib | 1425381-60-7 | 460.53 | 10mM | JAK; Syk |
T6145 | ZM39923 hydrochloride | 1021868-92-7 | 367.91 | 10mM | EGFR; JAK |
T8546 | BD750 | 892686-59-8 | 271.34 | 10mM | JAK; STAT |
T22338 | 2,6-Dichloro-N-(2-(cyclopropanecarboxamido)pyridin-4-yl)benzamide | 1258292-64-6 | 350.2 | 10mM | JAK |
T8719 | SC99 | 882290-02-0 | 336.15 | 10mM | Apoptosis; JAK; STAT |
T8742 | G5-7 | 939681-36-4 | 411.4 | 10mM | Apoptosis; JAK |
T4672 | Brevilin A | 16503-32-5 | 346.41 | 10mM | Anti-infection; Apoptosis; Autophagy; JAK; STAT |
T4657L | WHI-P97 HCl 211555-05-4(free base) | T4657L | 491.56 | 10mM | JAK |
TQ0037 | Abrocitinib | 1622902-68-4 | 323.41 | 10mM | JAK |
T12266 | Ilginatinib | 1239358-86-1 | 389.43 | 10mM | JAK; Tyrosine Kinases |
T10431 | Golidocitinib | 2091134-68-6 | 489.57 | 10mM | JAK |
T9195 | SHR0302 | 1445987-21-2 | 414.48 | 10mM | Apoptosis; JAK |
T21503 | (E/Z)-Zotiraciclib | 937270-47-8 | 372.46 | 10mM | CDK; FLT; JAK |
T15096 | Delgocitinib | 1263774-59-9 | 310.35 | 10mM | JAK; Tyrosine Kinases |
T9826 | GDC-0214 | 1831144-46-7 | 612.03 | 10mM | JAK |
T35900 | JAK2-IN-7 | 2593402-36-7 | 459.59 | 10mM | JAK |
TQ0010 | Brepocitinib | 1883299-62-4 | 389.4 | 10mM | JAK; Tyrosine Kinases |
T11710 | JAK-IN-5 | 2096999-92-5 | 474.57 | 10mM | JAK |
T39113L | Povorcitinib phosphate | 1637677-33-8 | 605.45 | 10mM | JAK |
T12549 | JAK-IN-11 | 916742-11-5 | 483.52 | 10mM | JAK |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |