HMGCR inhibitor kit 包含HMG-CoA 还原酶抑制剂,HMGCR 是体内催化胆固醇从头合成的关键酶,HMGCR 活性增高,肝脏合成胆固醇增多,可使胆汁中胆固醇饱和指数上升。抑制HMGCR 可降低TC、TG、LDI、VLDL 的血浆浓度,提高HDL 的血浆浓度,缓解多种疾病的进程。TargetMol 为您提供19种精选HMG-CoA 还原酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0672 | Pravastatin sodium | 81131-70-6 | 446.52 | 10mM | Autophagy; Ferroptosis; HMG-CoA Reductase |
T0683 | Mevastatin | 73573-88-3 | 390.51 | 10mM | Antibacterial; Antibiotic; Apoptosis; Autophagy; HMG-CoA Reductase; Lipid |
T0687 | Simvastatin | 79902-63-9 | 418.57 | 10mM | Apoptosis; Autophagy; Ferroptosis; HMG-CoA Reductase; Mitophagy |
T1207 | Lovastatin | 75330-75-5 | 404.54 | 10mM | Autophagy; Ferroptosis; HMG-CoA Reductase |
T1487 | Fluvastatin sodium | 93957-55-2 | 433.45 | 10mM | Autophagy; Ferroptosis; HMG-CoA Reductase |
T1510 | Rosuvastatin calcium | 147098-20-2 | 1001.14 | 10mM | Autophagy; HMG-CoA Reductase; Potassium Channel |
T1664 | Meglutol | 503-49-1 | 162.14 | 10mM | Autophagy; Endogenous Metabolite; HMG-CoA Reductase |
T1676 | Rosuvastatin | 287714-41-4 | 481.54 | 10mM | Autophagy; HMG-CoA Reductase; Potassium Channel |
T2534 | Pitavastatin calcium | 147526-32-7 | 880.98 | 10mM | Apoptosis; Autophagy; Endogenous Metabolite; HMG-CoA Reductase; Mitophagy |
T3116 | Atorvastatin hemicalcium salt | 134523-03-8 | 1155.34 | 10mM | Autophagy; Ferroptosis; HMG-CoA Reductase |
T3698 | alpha-Asarone | 2883-98-9 | 208.3 | 10mM | GABA Receptor; HMG-CoA Reductase; P450 |
T6450 | Clinofibrate | 30299-08-2 | 468.58 | 10mM | Autophagy; HMG-CoA Reductase |
T6994 | SR12813 | 126411-39-0 | 504.53 | 10mM | Autophagy; HMG-CoA Reductase |
T4717 | 25-Hydroxycholesterol | 2140-46-7 | 402.65 | 10mM | Endogenous Metabolite; HMG-CoA Reductase |
TN1733 | Hesperetin 7-O-glucoside | 31712-49-9 | 464.4 | 10mM | Anti-infection; Antibacterial; HMG-CoA Reductase |
T12092 | Monacolin J | 79952-42-4 | 320.42 | 10mM | Autophagy; HMG-CoA Reductase |
T14342 | Atorvastatin lactone | 125995-03-1 | 540.62 | 10mM | HMG-CoA Reductase |
T26644 | Apomine | 126411-13-0 | 562.66 | 10mM | HMG-CoA Reductase |
TN1438 | beta-Amyrin acetate | 1616-93-9 | 468.75 | 10mM | HMG-CoA Reductase;Antifungal;Epoxide Hydrolase;Antioxidant |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |