HIF/HIF-PH inhibitor/activator kit 包含缺氧诱导因子HIF/HIF 脯氨酰羟化酶HIF-PH 抑制剂/激活剂,HIF 是一种能够应答细胞内氧气浓度的降低而对多种基因进行调控的转录因子家族。HIF-PH 途径指的是通过HIF-PH 在氧分子的参与下使HIFα被快速降解的过程,在缺氧时可以调控体内的HIFα含量,从而调控血红细胞含量,改善贫血状况。TargetMol 为您提供34种精选HIF/HIF-PH 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1939 | DMOG | 89464-63-1 | 175.14 | 10mM | Autophagy; HIF; HIF/HIF Prolyl-Hydroxylase |
T2445 | FG-2216 | 223387-75-5 | 280.66 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T2488 | BAY 87-2243 | 1227158-85-1 | 525.53 | 10mM | Ferroptosis; HIF; HIF/HIF Prolyl-Hydroxylase |
T3169 | KC7F2 | 927822-86-4 | 570.38 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T3180 | JNJ-42041935 | 1193383-09-3 | 346.65 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T3494 | LW6 | 934593-90-5 | 435.52 | 10mM | Apoptosis; Dehydrogenase; HIF; HIF/HIF Prolyl-Hydroxylase |
T4106 | MK-8617 | 1187990-87-9 | 443.45 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T4381 | Lificiguat | 170632-47-0 | 304.34 | 10mM | Guanylate cyclase; HIF |
T6961 | PX-478 | 685898-44-6 | 394.12 | 10mM | Autophagy; HIF; HIF/HIF Prolyl-Hydroxylase |
T5176 | Desidustat | 1616690-16-4 | 332.31 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T5392 | TP0463518 | 1558021-37-6 | 431.83 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T5537 | IDF-11774 | 1429054-28-3 | 368.5 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T5684 | Ethyl 3,4-dihydroxybenzoate | 3943-89-3 | 182.17 | 10mM | Apoptosis; Autophagy; HIF/HIF Prolyl-Hydroxylase; NO Synthase; Reactive Oxygen Species |
T7692 | 2,4-DPD | 41438-38-4 | 223.23 | 10mM | HIF |
T7802 | M1001 | 874590-32-6 | 327.4 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T7880 | IOX4 | 1154097-71-8 | 328.33 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T7848 | PT-2385 | 1672665-49-4 | 383.34 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T15219 | Enarodustat | 1262132-81-9 | 340.33 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T13050 | SYP-5 | 1384268-04-5 | 312.38 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T12675L | PT2399 | 1672662-14-4 | 419.32 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T11561 | HIF-2α-IN-2 | 1672666-82-8 | 365.35 | 10mM | HIF; HIF/HIF Prolyl-Hydroxylase |
T001-00000002 | Izilendustat | 1303512-02-8 | 433.93 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T19832 | Acriflavine Hydrochloride | 8063-24-9 | 259.73 | 10mM | HIF |
T15396 | GN44028 | 1421448-26-1 | 305.33 | 10mM | HIF |
T9627 | PHD-1-IN-1 | 2009343-14-8 | 220.23 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T13398 | ZINC13466751 | 117953-17-0 | 363.41 | 10mM | HIF |
T16679 | Belzutifan | 1672668-24-4 | 383.34 | 10mM | HIF |
T9890 | HIF1-IN-3 | 333314-79-7 | 412.48 | 10mM | HIF |
T29797 | AKB-6899 | 1007377-55-0 | 290.25 | 10mM | HIF/HIF Prolyl-Hydroxylase;HIF;VEGFR |
T22022 | Adaptaquin | 385786-48-1 | 377.82 | 10mM | HIF |
T21653 | 1,4-DPCA | 331830-20-7 | 240.21 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T7836 | ML228 | 1357171-62-0 | 415.49 | 10mM | HIF |
T17105 | TM6089 | 863421-32-3 | 306.34 | 10mM | HIF/HIF Prolyl-Hydroxylase |
T36711 | FM19G11 | 329932-55-0 | 463.4 | 10mM | HIF |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |