GSK-3 inhibitor kit 包含 GSK-3抑制剂,GSK-3是一种非常保守的丝 Ser/Thr 激酶,参与肝糖的合成代谢,能作用于许多信号蛋白结构蛋白和转录因子,参与细胞分化、增殖、存活和凋亡的调控,常用于癌症、神经退行性疾病、神经精神类疾病等多种重大疾病的研究中。TargetMol 为您提供46种精选 GSK-3抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1260 | Cromolyn sodium | 15826-37-6 | 512.33 | 10mM | Calcium Channel; GSK-3; Potassium Channel |
T1741 | AZD1080 | 612487-72-6 | 334.37 | 10mM | GSK-3 |
T1755 | LY2090314 | 603288-22-8 | 512.53 | 10mM | GSK-3 |
T1778 | AT7519 Hydrochloride | 902135-91-5 | 418.71 | 10mM | Apoptosis; CDK; GSK-3 |
T1881 | AR-A014418 | 487021-52-3 | 308.31 | 10mM | GSK-3 |
T1917 | GSK 3 Inhibitor IX | 667463-62-9 | 356.17 | 10mM | Apoptosis; CDK; GSK-3; Tyrosine Kinases |
T1957 | AZD2858 | 486424-20-8 | 453.52 | 10mM | GSK-3 |
T1965 | Bikinin | 188011-69-0 | 273.08 | 10mM | GSK-3 |
T2166 | TWS119 | 601514-19-6 | 318.33 | 10mM | Autophagy; GSK-3 |
T2247 | KenPaullone | 142273-20-9 | 327.18 | 10mM | CDK; GSK-3 |
T2261 | IM-12 | 1129669-05-1 | 377.41 | 10mM | GSK-3 |
T2310 | CHIR-99021 | 252917-06-9 | 465.34 | 10mM | Autophagy; GSK-3; Wnt/beta-catenin |
T2378 | RGB-286638 free base | 784210-88-4 | 545.63 | 10mM | CDK; GSK-3; JAK; MEK |
T2608 | CHIR-98014 | 252935-94-7 | 486.31 | 10mM | FGFR; GSK-3; S6 Kinase; Src |
T3067 | Tideglusib | 865854-05-3 | 334.39 | 10mM | GSK-3 |
T3074 | CHIR 98024 | 556813-39-9 | 486.31 | 10mM | GSK-3; S6 Kinase |
T3077 | SB 216763 | 280744-09-4 | 371.22 | 10mM | Autophagy; GSK-3 |
T3385 | Gypenoside XVII | 80321-69-3 | 947.16 | 10mM | Endogenous Metabolite; Estrogen Receptor/ERR; GSK-3 |
T3684 | CP21R7 | 125314-13-8 | 317.3 | 10mM | GSK-3; PKC |
T6169 | Indirubin | 479-41-4 | 262.26 | 10mM | Apoptosis; CDK; GSK-3; Raf |
T6187 | TDZD-8 | 327036-89-5 | 222.26 | 10mM | GSK-3 |
T6206 | PHA-767491 | 845714-00-3 | 213.24 | 10mM | CDK; GSK-3 |
T6358 | 1-Azakenpaullone | 676596-65-9 | 328.16 | 10mM | GSK-3 |
T6659 | SB 415286 | 264218-23-7 | 359.72 | 10mM | Apoptosis; GSK-3 |
T6787 | BIO-acetoxime | 667463-85-6 | 398.21 | 10mM | Apoptosis; GSK-3; HSV |
T5200 | Indirubin-3'-monoxime | 160807-49-8 | 277.28 | 10mM | CDK; GSK-3; Lipoxygenase |
T5956 | VP3.15 dihydrobromide | 1281681-33-1 | 528.3 | 10mM | GSK-3; PDE |
T7473 | 5-Bromoindole | 10075-50-0 | 196.04 | 10mM | GSK-3 |
T7426 | Alsterpaullone | 237430-03-4 | 293.28 | 10mM | Apoptosis; CDK; GSK-3 |
T8605 | GS87 | 919936-70-2 | 337.36 | 10mM | GSK-3 |
T11467 | GSK-3β inhibitor 1 | 187325-53-7 | 222.24 | 10mM | GSK-3 |
T14066 | 9-ING-41 | 1034895-42-5 | 404.35 | 10mM | Apoptosis; Autophagy; GSK-3 |
T8908 | 4-Chloro-2'-bromoacetophenone | 536-38-9 | 233.49 | 10mM | GSK-3 |
T24111 | GSK3i XIII | 404828-08-6 | 301.35 | 10mM | GSK-3 |
T9025 | KY19382 | 2226664-93-1 | 360.2 | 10mM | GSK-3; Wnt/beta-catenin |
T10606 | BRD0705 | 2056261-41-5 | 321.42 | 10mM | GSK-3 |
T9138 | Indirubin-3′-oxime | 667463-82-3 | 277.28 | 10mM | CDK; GSK-3; JNK |
T9178 | (E/Z)-GSK-3β inhibitor 1 | 3367-88-2 | 222.24 | 10mM | GSK-3 |
T14072 | A-443654 | 552325-16-3 | 397.47 | 10mM | Akt; Casein Kinase; CDK; Chk; ERK; FLT; GSK-3; MAPK; PKA; PKC; S6 Kinase; Src; VEGFR |
T10202 | A 1070722 | 1384424-80-9 | 362.31 | 10mM | GSK-3 |
T9611 | PF-04802367 | 1962178-27-3 | 361.78 | 10mM | GSK-3 |
T9987 | WAY-352753 | 478482-74-5 | 303.77 | 10mM | GSK-3 |
T11960 | MBM-55 | 2083622-09-5 | 498.55 | 10mM | MAPK;S6 Kinase;DYRK;Chk;GSK-3;Bcr-Abl;Akt;Aurora Kinase;CDK |
T11471 | GSK-3β inhibitor 2 | 1702428-31-6 | 318.35 | 10mM | GSK-3 |
T11961 | MBM-55S | 2083624-07-9 | 734.73 | 10mM | MAPK;S6 Kinase;GSK-3;Bcr-Abl;CDK;CDK;Akt;Aurora Kinase |
T14613 | BIP-135 | 941575-71-9 | 421.24 | 10mM | GSK-3 |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |