FLT3 inhibitor kit 包含FMS 样酪氨酸激酶3 FLT3抑制剂,FLT3是一种Ⅲ型受体酪氨酸激酶,在造血细胞的存活、增殖和分化中起着重要作用。FLT3基因突变是急性髓系白血病患者常见的预后不良因素,突变型FLT3诱导多种细胞内信号通路的激活导致细胞增殖和抗凋亡,主要包括STAT5、MAPK 和AKT 等通路。TargetMol 为您提供47种精选FLT3抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0093L | Sorafenib | 284461-73-0 | 464.83 | 10mM | Apoptosis; Autophagy; c-Kit; Ferroptosis; FLT; PDGFR; Raf; VEGFR |
T1667 | Tandutinib | 387867-13-2 | 562.7 | 10mM | Apoptosis; c-Kit; CSF-1R; FLT; PDGFR; Src |
T1836 | AZD2932 | 883986-34-3 | 447.49 | 10mM | c-Kit; FLT; PDGFR; VEGFR |
T1938 | FLT3-IN-2 | 923562-23-6 | 416.83 | 10mM | FLT |
T1995 | Fedratinib | 936091-26-8 | 524.68 | 10mM | Apoptosis; c-RET; FLT; JAK |
T2051 | SKLB4771 | 1370256-78-2 | 537.66 | 10mM | FLT |
T2054 | Altiratinib | 1345847-93-9 | 510.46 | 10mM | c-Met/HGFR; FLT; Tie-2; Trk receptor; VEGFR |
T2066 | Quizartinib | 950769-58-1 | 560.67 | 10mM | Apoptosis; Autophagy; FLT; Ligands for Target Protein for PROTAC |
T2115 | Pexidartinib | 1029044-16-3 | 417.81 | 10mM | Apoptosis; c-Fms; c-Kit; CSF-1R; FLT |
T2272 | BPR1J-097 | 1327167-19-0 | 516.62 | 10mM | FLT |
T2341 | KW-2449 | 1000669-72-6 | 332.4 | 10mM | Apoptosis; Aurora Kinase; Bcr-Abl; c-Kit; FGFR; FLT; JAK; Src |
T2358 | ENMD-2076 | 934353-76-1 | 375.47 | 10mM | Apoptosis; Aurora Kinase; c-RET; FGFR; FLT; PDGFR; Src; VEGFR |
T2514 | Linifanib | 796967-16-3 | 375.4 | 10mM | Apoptosis; Autophagy; c-Fms; c-Kit; CSF-1R; FLT; PDGFR; VEGFR |
T2516 | Amuvatinib | 850879-09-3 | 447.51 | 10mM | Apoptosis; c-Kit; c-Met/HGFR; c-RET; DNA/RNA Synthesis; FLT; PDGFR |
T2586 | Cabozantinib | 849217-68-1 | 501.5 | 10mM | Apoptosis; c-Kit; c-Met/HGFR; c-RET; FLT; TAM Receptor; VEGFR |
T2620 | G-749 | 1457983-28-6 | 521.41 | 10mM | Apoptosis; Aurora Kinase; c-RET; FLT; TAM Receptor |
T2638 | Gandotinib | 1229236-86-5 | 469.94 | 10mM | FGFR; FLT; JAK; VEGFR |
T2677 | Crenolanib | 670220-88-9 | 443.54 | 10mM | Autophagy; FLT; PDGFR |
T3065 | TG101209 | 936091-14-4 | 509.67 | 10mM | Apoptosis; Autophagy; c-RET; FLT; JAK |
T3068 | AT9283 | 896466-04-9 | 381.43 | 10mM | Apoptosis; Aurora Kinase; Autophagy; Bcr-Abl; FLT; JAK |
T3078 | SGI-1776 | 1025065-69-3 | 405.42 | 10mM | Apoptosis; Autophagy; FLT; Pim |
T4053 | AST 487 | 630124-46-8 | 529.56 | 10mM | Bcr-Abl; c-Kit; c-RET; FLT; VEGFR |
T4209 | TAK-659 hydrochloride | 1952251-28-3 | 380.85 | 10mM | FLT; JAK; Syk; Tyrosine Kinases; VEGFR |
T4227 | SB1317 hydrochloride (1204918-72-8(free base)) | T4227 | 408.92 | 10mM | CDK; FLT; JAK |
T4409 | Gilteritinib | 1254053-43-4 | 552.72 | 10mM | c-Kit; FLT; TAM Receptor |
T4419 | UNC2025 2HCl (1429881-91-3(free base)) | T4419 | 549.62 | 10mM | FLT; TAM Receptor |
T6020 | Pacritinib | 937272-79-2 | 472.58 | 10mM | FLT; JAK; Tyrosine Kinases |
T6138 | TCS 359 | 301305-73-7 | 360.43 | 10mM | FLT |
T6174 | R406 | 841290-81-1 | 628.63 | 10mM | Apoptosis; FLT; Syk |
T6479 | Dovitinib lactate hydrate | 915769-50-5 | 482.51 | 10mM | c-Kit; FGFR; FLT; PDGFR; VEGFR |
T6756 | AMG 925 | 1401033-86-0 | 471.55 | 10mM | CDK; FLT |
T7007 | UNC2025 | 1429881-91-3 | 476.7 | 10mM | FLT; TAM Receptor |
T6S0033 | Crotonoside | 1818-71-9 | 283.24 | 10mM | FLT; HDAC |
T7673 | ATH686 | 853299-52-2 | 515.53 | 10mM | Apoptosis; FLT |
T8317 | 5'-Fluoroindirubinoxime | 861214-33-7 | 295.27 | 10mM | FLT |
T8326 | BMS-2 | 888719-03-7 | 458.42 | 10mM | c-Met/HGFR; FLT; VEGFR |
T16144 | MRX-2843 | 1429882-07-4 | 488.67 | 10mM | FLT |
T9027 | CA-4948 | 1801344-14-8 | 491.5 | 10mM | FLT; IRAK |
T9017 | HPK1-IN-2 | 2056122-11-1 | 380.47 | 10mM | FLT; Src |
T11298 | FLT3-IN-3 | 2229050-90-0 | 490.64 | 10mM | FLT |
TQ0235 | AC710 | 1351522-04-7 | 562.7 | 10mM | c-Kit; FLT; PDGFR |
T13564 | AZ7550 | 1421373-99-0 | 485.58 | 10mM | ACK; ALK; BTK; Drug Metabolite; EGFR; FAK; FLT; IGF-1R; MLK; MNK; PYK2; Tyrosine Kinases |
T9428 | HM43239 | 2569527-64-4 | 501.07 | 10mM | FLT |
T9473 | 4SC-203 | 895533-09-2 | 642.77 | 10mM | FLT |
T21503 | (E/Z)-Zotiraciclib | 937270-47-8 | 372.46 | 10mM | CDK; FLT; JAK |
T38562 | AKN-028 | 1175017-90-9 | 302.33 | 10mM | FLT |
T9856 | FLT3-IN-10 | 2088735-51-5 | 254.26 | 10mM | FLT |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |