FGFR inhibitor kit 包含成纤维细胞生长因子受体 FGFR 抑制剂,FGFR 属于受体激酶家族,包括四种受体亚型(FGFR-1,2,3 和4)及一些异构分子,通过与成纤维细胞生长因子形成三元复合物参与调节生物的生理过程,如胚胎发育,伤口愈合和血管生成等。TargetMol 为您提供52种精选FGFR 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0097L | Pazopanib | 444731-52-6 | 437.52 | 10mM | Autophagy; c-Kit; FGFR; PDGFR; VEGFR |
T0724 | Formononetin | 485-72-3 | 268.27 | 10mM | Apoptosis; FGFR |
T1777 | Nintedanib | 656247-17-5 | 539.62 | 10mM | FGFR; FLT; PDGFR; Src; VEGFR |
T1886 | TAK-632 | 1228591-30-7 | 554.52 | 10mM | Aurora Kinase; FGFR; PDGFR; Raf |
T1895 | SKLB 610 | 1125780-41-7 | 415.37 | 10mM | FGFR; PDGFR; VEGFR |
T1948 | AZD4547 | 1035270-39-3 | 463.57 | 10mM | FGFR; VEGFR |
T1975 | Infigratinib | 872511-34-7 | 560.48 | 10mM | Apoptosis; FGFR |
T2094 | Danusertib | 827318-97-8 | 474.55 | 10mM | Aurora Kinase; Autophagy; Bcr-Abl; c-RET; FGFR; Trk receptor |
T2215 | Ferulic Acid | 1135-24-6 | 194.19 | 10mM | Endogenous Metabolite; FGFR |
T2347 | BLU9931 | 1538604-68-0 | 509.38 | 10mM | FGFR |
T2358 | ENMD-2076 | 934353-76-1 | 375.47 | 10mM | Apoptosis; Aurora Kinase; c-RET; FGFR; FLT; PDGFR; Src; VEGFR |
T2361 | LY2874455 | 1254473-64-7 | 444.31 | 10mM | FGFR; VEGFR |
T2372 | Ponatinib | 943319-70-8 | 532.56 | 10mM | Autophagy; Bcr-Abl; c-Kit; FGFR; PDGFR; Src; VEGFR |
T2638 | Gandotinib | 1229236-86-5 | 469.94 | 10mM | FGFR; FLT; JAK; VEGFR |
T2642 | PD173074 | 219580-11-7 | 523.67 | 10mM | Apoptosis; EGFR; FGFR; IGF-1R; Src; VEGFR |
T2857 | 2,5-Dihydroxybenzoic acid | 490-79-9 | 154.12 | 10mM | Endogenous Metabolite; FGFR |
T3274 | S49076 | 1265965-22-7 | 438.13 | 10mM | c-Met/HGFR; FGFR; TAM Receptor |
T3456 | Fisogatinib | 1707289-21-1 | 503.38 | 10mM | FGFR |
T3466 | FIIN-3 | 1637735-84-2 | 691.61 | 10mM | EGFR; FGFR |
T3492 | PD-166866 | 192705-79-6 | 396.45 | 10mM | Autophagy; FGFR |
T3726 | Erdafitinib | 1346242-81-6 | 446.55 | 10mM | Apoptosis; FGFR |
T4235 | Roblitinib | 1708971-55-4 | 506.57 | 10mM | FGFR |
T4318 | EOC317 | 939805-30-8 | 591.54 | 10mM | FGFR; Tie-2; VEGFR |
T6024 | Zoligratinib | 1265229-25-1 | 356.38 | 10mM | FGFR |
T6082 | SSR128129E | 848318-25-2 | 346.31 | 10mM | FGFR |
T6184 | Orantinib | 252916-29-3 | 310.35 | 10mM | Apoptosis; FGFR; PDGFR; VEGFR |
T6479 | Dovitinib lactate hydrate | 915769-50-5 | 482.51 | 10mM | c-Kit; FGFR; FLT; PDGFR; VEGFR |
T6836 | FIIN-2 | 1633044-56-0 | 634.73 | 10mM | FGFR |
T6920 | ON123300 | 1357470-29-1 | 429.52 | 10mM | AMPK; c-RET; CDK; FGFR; JAK; PDGFR; Src |
T6996 | SU 5402 | 215543-92-3 | 296.32 | 10mM | FGFR; PDGFR; VEGFR |
T2S0007 | Ferulic acid sodium | 24276-84-4 | 216.16 | 10mM | 5-HT Receptor; Endogenous Metabolite; FGFR; Reactive Oxygen Species |
T5044 | Futibatinib | 1448169-71-8 | 418.45 | 10mM | FGFR |
T5001 | Nintedanib esylate | 656247-18-6 | 649.76 | 10mM | FGFR; PDGFR; VEGFR |
T5122 | Alofanib | 1612888-66-0 | 413.4 | 10mM | Apoptosis; FGFR |
T5466 | Tyrosine kinase-IN-1 | 705946-27-6 | 445.54 | 10mM | FGFR; FLT; PDGFR; VEGFR |
T5473 | ASP5878 | 1453208-66-6 | 407.38 | 10mM | FGFR |
T7611 | ODM-203 | 1430723-35-5 | 505.54 | 10mM | FGFR; VEGFR |
T7738 | H3B-6527 | 1702259-66-2 | 629.53 | 10mM | FGFR |
T8541 | Lenvatinib mesylate | 857890-39-2 | 522.96 | 10mM | c-Kit; c-RET; FGFR; PDGFR; VEGFR |
TQ0228 | Derazantinib | 1234356-69-4 | 468.57 | 10mM | FGFR |
T12401 | Pemigatinib | 1513857-77-6 | 487.5 | 10mM | FGFR |
TQ0015 | PRN1371 | 1802929-43-6 | 561.46 | 10mM | c-Fms; CSF-1R; FGFR |
T22306 | DGY-06-116 | T22306 | 597.11 | 10mM | FGFR; Src |
T11279 | FGFR1/DDR2 inhibitor 1 | 2308497-58-5 | 501.5 | 10mM | Discoidin Domain Receptor (DDR); FGFR |
T8976 | PD-089828 | 179343-17-0 | 405.28 | 10mM | EGFR; FGFR; PDGFR; Src |
T9030 | SU4984 | 186610-89-9 | 333.38 | 10mM | FGFR; IGF-1R; PDGFR |
T15185 | Lucitanib | 1058137-23-7 | 443.49 | 10mM | FGFR; VEGFR |
TQ0256 | FGFR4-IN-1 | 1708971-72-5 | 493.52 | 10mM | FGFR |
T23127 | PD-161570 | 192705-80-9 | 532.51 | 10mM | EGFR; FGFR; PDGFR; Src |
TQ0317 | R1530 | 882531-87-5 | 356.78 | 10mM | FGFR; FLT; PDGFR; VEGFR |
T13824 | PP58 | 212391-58-7 | 456.33 | 10mM | PDGFR;FGFR;Src;p38 MAPK;TNF |
T60185 | FGFR2-IN-3 | 2549174-42-5 | 509.53 | 10mM | FGFR |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |