ER stress pathway inhibitor/inducer kit 包含内质网ER 应激抑制剂/诱导剂,内质网应激是由多种应激源引起的,如内质网腔内错误折叠蛋白的积累、营养剥夺、缺氧、治疗药物和炎症因子,参与神经退行性疾病、缺血再灌注损伤、糖尿病、肿瘤等多种疾病。TargetMol 为您提供45种精选ER 应激抑制剂/诱导剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0012 | Cinchonine | 118-10-5 | 294.39 | 10mM | Apoptosis; P-gp; Parasite |
T0772 | Troxerutin | 7085-55-4 | 742.67 | 10mM | NOD-like Receptor (NLR) |
T1535 | Sodium 4-phenylbutyrate | 1716-12-7 | 186.18 | 10mM | Apoptosis; Autophagy; HDAC |
T1742 | 4E1rcat | 328998-25-0 | 478.45 | 10mM | Autophagy; PERK |
T1862 | PR-619 | 2645-32-1 | 223.33 | 10mM | Apoptosis; Autophagy; DUB |
T2417 | Sal003 | 1164470-53-4 | 463.21 | 10mM | Apoptosis; PERK; Phosphatase |
T2614 | GSK2606414 | 1337531-36-8 | 451.44 | 10mM | Apoptosis; Autophagy; PERK |
T2665 | 4EGI-1 | 315706-13-9 | 451.28 | 10mM | Apoptosis; Autophagy; PERK |
T3045 | Salubrinal | 405060-95-9 | 479.81 | 10mM | Apoptosis; Autophagy; HSV; PERK; Phosphatase |
T3207 | Briciclib | 865783-99-9 | 474.42 | 10mM | Autophagy; CDK; PERK |
T3395 | Timosaponin AIII | 41059-79-4 | 740.92 | 10mM | AChE; mTOR |
T3427 | Polydatin | 27208-80-6 | 390.39 | 10mM | Apoptosis; Autophagy; Mitophagy; NF-κB |
T3780 | Oroxin B | 114482-86-9 | 594.52 | 10mM | Antioxidant; Apoptosis; Autophagy; PI3K; PTEN |
T4304 | Azoramide | 932986-18-0 | 308.82 | 10mM | Apoptosis; PERK |
T6183 | ISRIB (trans-isomer) | 1597403-47-8 | 451.34 | 10mM | Apoptosis; Autophagy; PERK |
T6800 | CCF642 | 346640-08-2 | 378.45 | 10mM | Others |
T6886 | MCB-613 | 1162656-22-5 | 304.39 | 10mM | Src |
T6993 | Tauroursodeoxycholate sodium | 35807-85-3 | 521.69 | 10mM | Apoptosis; Caspase; ERK |
T5A2461 | Bufotalin | 471-95-4 | 444.56 | 10mM | Apoptosis; Reactive Oxygen Species |
T6S1292 | Levistolide A | 88182-33-6 | 380.48 | 10mM | Apoptosis |
T5173 | SBI-0640756 | 1821280-29-8 | 404.82 | 10mM | Autophagy; PERK |
T5886 | 4-Phenylbutyric acid | 1821-12-1 | 164.2 | 10mM | HDAC; Virus Protease |
T7150 | BTdCPU | 1257423-87-2 | 339.2 | 10mM | Apoptosis; PERK; Phosphatase |
T7127 | DC260126 | 346692-04-4 | 307.38 | 10mM | Apoptosis; GPR |
T7955 | EB-3D | 1839150-63-8 | 644.4 | 10mM | AChR; AMPK; Apoptosis |
T8464 | RA-9 | 919091-63-7 | 365.34 | 10mM | Apoptosis; DUB |
T14080 | AA147 | 393121-74-9 | 255.31 | 10mM | Others |
T16974 | TAK-243 | 1450833-55-2 | 519.52 | 10mM | Apoptosis; E1/E2/E3 Enzyme; NF-κB |
T8901 | YUM70 | 423145-35-1 | 398.84 | 10mM | Apoptosis; GPR; HSP |
TN1702 | Glycycoumarin | 94805-82-0 | 368.37 | 10mM | Autophagy; JNK; P450 |
TN1586 | Dihydrorotenone | 6659-45-6 | 396.43 | 10mM | Apoptosis; Mitochondrial Metabolism |
T8982 | RH01687 | 302901-13-9 | 336.75 | 10mM | Others |
TN2225 | Soyasapogenol B | 595-15-3 | 458.7 | 10mM | Apoptosis; Autophagy |
T9110 | Ceapin-A7 | 2323027-38-7 | 470.32 | 10mM | Others |
T2930 | α-Lipoic Acid | 62-46-4 | 206.32 | 10mM | Endogenous Metabolite; HIV Protease; Mitochondrial Metabolism; NF-κB |
T29017 | TrxR1-IN-B19 | 170950-29-5 | 354.4 | 10mM | Others |
T9149 | 2BAct | 2143542-28-1 | 440.8 | 10mM | PERK |
T3564 | SHP099 | 1801747-42-1 | 352.26 | 10mM | PERK; Phosphatase |
T24855 | TASIN-1 Hydrochloride | 1678515-13-3 | 388.95 | 10mM | APC |
T13416 | ZX-29 | 2254805-62-2 | 518.03 | 10mM | ALK |
T14044 | 4E2RCat | 432499-63-3 | 455.93 | 10mM | PERK |
T20797 | NE-100 hydrochloride | 149409-57-4 | 391.98 | 10mM | Sigma receptor |
T9564 | IRE1α kinase-IN-1 | 2328097-41-0 | 504.99 | 10mM | IRE1 |
T40130 | Nur77 modulator 1 | 2469975-55-9 | 495.6 | 10mM | Others |
T27579 | ICL-CCIC-0019 | 936498-64-5 | 572.46 | 10mM | AChR |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |