Endothelin Receptor antagonist kit 包含内皮素受体拮抗剂,内皮素具有强烈缩血管作用,诱导血管生成、促分化、促细胞有丝分裂和类细胞生长因子。内皮素还有强大的正性肌力作用,反射性引起心率抑制,造成心肌供血不足.而且还可诱发心肌细胞糖超载,心律失常以及心肌能量代谢障碍。内皮素受体拮抗剂常用于心绞痛、AMI、心肌1/R 损伤、缺血性心脏病的防治研究。TargetMol 为您提供18种精选内皮素受体拮抗剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0750 | Sulfisoxazole | 127-69-5 | 267.31 | 10mM | Antibacterial; Antibiotic; Autophagy; Endothelin Receptor |
T1655 | Ambrisentan | 177036-94-1 | 378.42 | 10mM | Endothelin Receptor |
T2561 | Macitentan | 441798-33-0 | 588.27 | 10mM | Apoptosis; Endothelin Receptor |
T3194 | Ro 46-2005 | 150725-87-4 | 473.54 | 10mM | Endothelin Receptor |
T3474 | RO 46-8443 | 175556-12-4 | 609.69 | 10mM | Endothelin Receptor |
T6264 | Bosentan | 147536-97-8 | 551.61 | 10mM | Endothelin Receptor |
T6265 | Bosentan (hydrate) | 157212-55-0 | 569.63 | 10mM | Endothelin Receptor |
T6672 | Sitaxsentan sodium | 210421-74-2 | 476.89 | 10mM | Endothelin Receptor |
T6792 | BQ-123 | 136553-81-6 | 610.7 | 10mM | Endothelin Receptor |
T5458 | Darusentan | 171714-84-4 | 410.43 | 10mM | Endothelin Receptor |
T7817 | Aprocitentan | 1103522-45-7 | 546.19 | 10mM | Endothelin Receptor |
T5355 | Sparsentan | 254740-64-2 | 592.8 | 10mM | Endothelin Receptor; RAAS |
T21790 | BMS 182874 hydrochloride | 1215703-04-0 | 381.88 | 10mM | Endothelin Receptor |
TQ0259 | Atrasentan | 173937-91-2 | 510.62 | 10mM | Endothelin Receptor |
TQ0282 | Avosentan | 290815-26-8 | 479.51 | 10mM | Endothelin Receptor |
TQ0270 | Atrasentan hydrochloride | 195733-43-8 | 547.08 | 10mM | Endothelin Receptor |
TP1219 | Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate | 1366000-58-9 | 3140.5 | 10mM | Endothelin Receptor |
T15596 | IRL 2500 | 169545-27-1 | 573.68 | 10mM | Endothelin Receptor |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |