DHFR inhibitor kit 包含二氢叶酸还原酶 DHFR 抑制剂,DHFR 是一类利用 NADPH 为辅因子催化二氢叶酸还原成四氢叶酸的胞浆蛋白酶类,在机体细胞一碳单位转运、胸腺嘧啶合成以及 DNA 合成中发挥重要作用。DHFR 抑制剂可抑制 DNA 的合成,导致细胞死亡,常用于恶性肿瘤的治疗研究。TargetMol 为您提供13种精选 DHFR 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0189 | Pemetrexed | 137281-23-3 | 427.41 | 10 mM | Antifolate; Autophagy; DHFR; DNA/RNA Synthesis |
T0189L | Pemetrexed disodium | 150399-23-8 | 471.37 | 10 mM | Antifolate; Apoptosis; Autophagy; DHFR; DNA/RNA Synthesis |
T0849 | Pyrimethamine | 58-14-0 | 248.71 | 10 mM | Antifolate; DHFR; Parasite |
T1153 | Trimethoprim | 738-70-5 | 290.32 | 10 mM | Antibacterial; Antibiotic; Antifolate; DHFR; DNA/RNA Synthesis |
T2204 | Diaveridine | 5355-16-8 | 260.29 | 10 mM | Antibacterial; Antifolate; DHFR |
T6120 | Pralatrexate | 146464-95-1 | 477.47 | 10 mM | Antifolate; Apoptosis; DHFR; TAM Receptor |
T6226 | Pemetrexed disodium hemipenta hydrate | 357166-30-4 | 518.43 | 10 mM | Antifolate; Apoptosis; Autophagy; DHFR; DNA/RNA Synthesis |
T36692 | Fanotaprim | 2120282-75-7 | 378.43 | 10 mM | DHFR |
T1485 | Methotrexate | 59-05-2 | 454.44 | 10 mM | ADC Cytotoxin; Antifolate; Apoptosis; Dehydrogenase; DNA/RNA Synthesis |
T4382 | Proguanil hydrochloride | 637-32-1 | 290.19 | 10 mM | Antifolate; Dehydrogenase; DNA/RNA Synthesis; Parasite |
T7730 | Aminopterin | 54-62-6 | 440.41 | 10 mM | Antifolate |
T8003 | Methotrexate disodium | 7413-34-5 | 498.4 | 10 mM | ADC Cytotoxin; Antifolate; Apoptosis; Dehydrogenase; DNA/RNA Synthesis |
T8548 | Metoprine | 7761-45-7 | 269.13 | 10 mM | Antifolate; Histamine Receptor; Histone Methyltransferase |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |