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DHFR inhibitor kit

DHFR inhibitor kit

现 货
产品编号 CL0132 DHFR inhibitor kit
  库化合物信息   Excel SDF

DHFR inhibitor kit 包含二氢叶酸还原酶 DHFR 抑制剂,DHFR 是一类利用 NADPH 为辅因子催化二氢叶酸还原成四氢叶酸的胞浆蛋白酶类,在机体细胞一碳单位转运、胸腺嘧啶合成以及 DNA 合成中发挥重要作用。DHFR 抑制剂可抑制 DNA 的合成,导致细胞死亡,常用于恶性肿瘤的治疗研究。TargetMol 为您提供13种精选 DHFR 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
规格
10 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品组成

ID Compound CAS MW Concentration Target
T0189 Pemetrexed 137281-23-3 427.41 10 mM Antifolate; Autophagy; DHFR; DNA/RNA Synthesis
T0189L Pemetrexed disodium 150399-23-8 471.37 10 mM Antifolate; Apoptosis; Autophagy; DHFR; DNA/RNA Synthesis
T0849 Pyrimethamine 58-14-0 248.71 10 mM Antifolate; DHFR; Parasite
T1153 Trimethoprim 738-70-5 290.32 10 mM Antibacterial; Antibiotic; Antifolate; DHFR; DNA/RNA Synthesis
T2204 Diaveridine 5355-16-8 260.29 10 mM Antibacterial; Antifolate; DHFR
T6120 Pralatrexate 146464-95-1 477.47 10 mM Antifolate; Apoptosis; DHFR; TAM Receptor
T6226 Pemetrexed disodium hemipenta hydrate 357166-30-4 518.43 10 mM Antifolate; Apoptosis; Autophagy; DHFR; DNA/RNA Synthesis
T36692 Fanotaprim 2120282-75-7 378.43 10 mM DHFR
T1485 Methotrexate 59-05-2 454.44 10 mM ADC Cytotoxin; Antifolate; Apoptosis; Dehydrogenase; DNA/RNA Synthesis
T4382 Proguanil hydrochloride 637-32-1 290.19 10 mM Antifolate; Dehydrogenase; DNA/RNA Synthesis; Parasite
T7730 Aminopterin 54-62-6 440.41 10 mM Antifolate
T8003 Methotrexate disodium 7413-34-5 498.4 10 mM ADC Cytotoxin; Antifolate; Apoptosis; Dehydrogenase; DNA/RNA Synthesis
T8548 Metoprine 7761-45-7 269.13 10 mM Antifolate; Histamine Receptor; Histone Methyltransferase

化合物库定制

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包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (CL0132)
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化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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