Casein Kinase inhibitor kit 包含酪蛋白激酶抑制剂,酪蛋白激酶催化肽链中邻近酸性氨基酸残基的丝氨酸/苏氨酸磷酸化的酶,主要包括酪蛋白激酶1和酪蛋白激酶2,在细胞分裂与凋亡、DNA 修复、P53调控、周期性节律等多种机体生理活动中发挥重要作用。TargetMol 为您提供32种精选酪蛋白激酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0465 | Ellagic acid | 476-66-4 | 302.19 | 10mM | Carbonic Anhydrase; Casein Kinase; Endogenous Metabolite; Hedgehog/Smoothened; PKA; PKC; Reactive Oxygen Species; Syk; Topoisomerase |
T1828 | TTP 22 | 329907-28-0 | 330.42 | 10mM | Casein Kinase |
T1877 | LH846 | 639052-78-1 | 316.81 | 10mM | Casein Kinase |
T2008 | LY294002 | 154447-36-6 | 307.34 | 10mM | Apoptosis; Autophagy; Casein Kinase; DNA-PK; PI3K |
T2048 | LY-364947 | 396129-53-6 | 272.3 | 10mM | Casein Kinase; MLK; RIP kinase; TGF-beta/Smad |
T2259 | Silmitasertib | 1009820-21-6 | 349.77 | 10mM | Autophagy; Casein Kinase |
T2440 | IC261 | 186611-52-9 | 311.33 | 10mM | Apoptosis; Casein Kinase; CDK |
T2449 | D4476 | 301836-43-1 | 398.41 | 10mM | ALK; Apoptosis; Autophagy; Casein Kinase |
T2695 | TBB | 17374-26-4 | 434.71 | 10mM | Casein Kinase; CDK; GSK-3 |
T2702 | IWP-2 | 686770-61-6 | 466.6 | 10mM | Casein Kinase; Porcupine; Wnt/beta-catenin |
T2869 | Emodin | 518-82-1 | 270.24 | 10mM | Autophagy; Casein Kinase; SARS-CoV |
T3073 | PF-670462 | 950912-80-8 | 410.32 | 10mM | Casein Kinase |
T3972 | SR-3029 | 1454585-06-8 | 480.45 | 10mM | Casein Kinase |
T6150 | TAK-715 | 303162-79-0 | 399.51 | 10mM | Casein Kinase; JNK; p38 MAPK |
T6735 | XL413 hydrochloride | 1169562-71-3 | 326.18 | 10mM | Casein Kinase; CDK; Pim |
T4645 | TA-01 | 1784751-18-3 | 351.32 | 10mM | Autophagy; Casein Kinase; p38 MAPK |
T5056 | PF-4800567 | 1188296-52-7 | 359.8 | 10mM | Casein Kinase |
T5358 | Longdaysin | 1353867-91-0 | 335.33 | 10mM | Casein Kinase; CDK; ERK |
T5393 | CK1-IN-1 | 1784751-20-7 | 383.39 | 10mM | Casein Kinase; p38 MAPK |
T7390 | DMAT | 749234-11-5 | 476.79 | 10mM | Casein Kinase |
T15024 | Silmitasertib sodium salt | 1309357-15-0 | 371.75 | 10mM | Autophagy; Casein Kinase |
T14069 | A-3 hydrochloride | 78957-85-4 | 321.22 | 10mM | CaMK; Casein Kinase; PKA; PKC |
T8987 | Epiblastin A | 16470-02-3 | 287.71 | 10mM | Casein Kinase |
T7949 | NCC007 | 2342583-66-6 | 447.5 | 10mM | Casein Kinase |
T9356 | (E/Z)-GO289 | 694522-87-7 | 419.3 | 10mM | Casein Kinase |
T19913 | CKI-7 | 1177141-67-1 | 358.67 | 10mM | Casein Kinase; CDK; ROCK; S6 Kinase; SGK |
T35557 | CK2 inhibitor 2 | 2641079-92-5 | 392.84 | 10mM | Casein Kinase |
T60005 | WAY-296817 | 349438-74-0 | 328.39 | 10mM | Casein Kinase |
T10547 | BioE-1115 | 1268863-35-9 | 339.36 | 10mM | Casein Kinase;Serine/threonin kinase |
T21915 | TBCA | 934358-00-6 | 463.74 | 10mM | Casein Kinase |
T10827 | CK2/ERK8-IN-1 | 1085822-09-8 | 534.82 | 10mM | Casein Kinase;ERK;Pim;DYRK;Apoptosis |
T60067 | WAY-297174 | 442571-27-9 | 268.36 | 10mM | Casein Kinase |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |