Aurora Kinase inhibitor kit 包含极光激酶抑制剂,极光激酶对细胞有丝分裂以及肿瘤形成很重要,参与了中心体成熟分离、纺锤体组装维持、染色体分离和胞质分裂等活动,不正常的有丝分裂过程可能导致癌变或凋亡。TargetMol 为您提供39种精选极光激酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1825 | Reversine | 656820-32-5 | 393.49 | 10mM | Adenosine Receptor; Aurora Kinase; Autophagy |
T1886 | TAK-632 | 1228591-30-7 | 554.52 | 10mM | Aurora Kinase; FGFR; PDGFR; Raf |
T2094 | Danusertib | 827318-97-8 | 474.55 | 10mM | Aurora Kinase; Autophagy; Bcr-Abl; c-RET; FGFR; Trk receptor |
T2241 | Alisertib | 1028486-01-2 | 518.92 | 10mM | Apoptosis; Aurora Kinase; Autophagy |
T2341 | KW-2449 | 1000669-72-6 | 332.4 | 10mM | Apoptosis; Aurora Kinase; Bcr-Abl; c-Kit; FGFR; FLT; JAK; Src |
T2358 | ENMD-2076 | 934353-76-1 | 375.47 | 10mM | Apoptosis; Aurora Kinase; c-RET; FGFR; FLT; PDGFR; Src; VEGFR |
T2471 | MK-8745 | 885325-71-3 | 431.91 | 10mM | Apoptosis; Aurora Kinase |
T2509 | Tozasertib | 639089-54-6 | 464.59 | 10mM | Aurora Kinase; Autophagy |
T2602 | Barasertib-HQPA | 722544-51-6 | 507.56 | 10mM | Apoptosis; Aurora Kinase |
T2611 | CCT 137690 | 1095382-05-0 | 551.48 | 10mM | Apoptosis; Aurora Kinase |
T2617 | SNS-314 Mesylate | 1146618-41-8 | 527.04 | 10mM | Aurora Kinase |
T2620 | G-749 | 1457983-28-6 | 521.41 | 10mM | Apoptosis; Aurora Kinase; c-RET; FLT; TAM Receptor |
T2709 | TAK-901 | 934541-31-8 | 504.64 | 10mM | Aurora Kinase; CDK; JAK; Src |
T3068 | AT9283 | 896466-04-9 | 381.43 | 10mM | Apoptosis; Aurora Kinase; Autophagy; Bcr-Abl; FLT; JAK |
T3109 | SP600125 | 129-56-6 | 220.23 | 10mM | Apoptosis; Aurora Kinase; Autophagy; Ferroptosis; JNK; Trk receptor |
T6028 | PF 477736 | 952021-60-2 | 419.48 | 10mM | Aurora Kinase; c-Fms; c-RET; CDK; Chk; FGFR; FLT; Src; VEGFR |
T6057 | URMC-099 | 1229582-33-5 | 421.54 | 10mM | Aurora Kinase; Autophagy; Bcr-Abl; c-Met/HGFR; CDK; DNA Alkylation; IGF-1R; LRRK2; MEK; MLK; ROCK; SGK; Src; Syk; Trk receptor; VEGFR |
T6077 | ZM-447439 | 331771-20-1 | 513.59 | 10mM | Apoptosis; Aurora Kinase; MEK; Src |
T6126 | JNJ-7706621 | 443797-96-4 | 394.36 | 10mM | Apoptosis; Aurora Kinase; CDK |
T6315 | MLN8054 | 869363-13-3 | 476.86 | 10mM | Aurora Kinase; Casein Kinase; PKA; Src |
T6338 | PHA-680632 | 398493-79-3 | 501.62 | 10mM | Aurora Kinase; FGFR; PLK |
T6380 | AMG 900 | 945595-80-2 | 503.58 | 10mM | Aurora Kinase; p38 MAPK; Tyrosine Kinases |
T6458 | CYC-116 | 693228-63-6 | 368.46 | 10mM | Aurora Kinase; CDK; FLT; S6 Kinase; VEGFR |
T6532 | Hesperadin | 422513-13-1 | 516.65 | 10mM | Aurora Kinase; Autophagy; Influenza Virus; Parasite |
T6767 | TCS7010 | 1158838-45-9 | 588.07 | 10mM | Apoptosis; Aurora Kinase |
T6785 | BI-847325 | 1207293-36-4 | 464.56 | 10mM | Apoptosis; Aurora Kinase; MEK |
T5524 | Aurora kinase inhibitor-3 | 879127-16-9 | 413.4 | 10mM | Aurora Kinase |
T8685 | SP-146 | T8685 | 453.47 | 10mM | Aurora Kinase |
T8866 | GW779439X | 551919-98-3 | 454.45 | 10mM | Antibacterial; Apoptosis; Aurora Kinase; CDK |
T21981 | Phthalazinone pyrazole | 880487-62-7 | 317.34 | 10mM | Aurora Kinase |
T16359 | NU6140 | 444723-13-1 | 422.52 | 10mM | Aurora Kinase; CDK |
T9040 | Aurora kinase inhibitor-2 | 331770-21-9 | 400.43 | 10mM | Aurora Kinase |
T14927 | Centrinone | 1798871-30-3 | 633.65 | 10mM | Aurora Kinase; PLK |
T17267 | XL228 | 898280-07-4 | 437.54 | 10mM | Aurora Kinase; Bcr-Abl; IGF-1R; Src |
T001-00000005 | AKI603 | 1432515-73-5 | 409.45 | 10mM | Aurora Kinase |
T22012 | 7BIO | 916440-85-2 | 356.17 | 10mM | Aurora Kinase; DYRK; FLT |
T10215 | AAPK-25 | 2247919-28-2 | 442.32 | 10mM | Aurora Kinase;PLK;Apoptosis |
T41256 | SP-96 | 2682114-54-9 | 453.47 | 10mM | Aurora Kinase |
T35570 | Chiauranib | 1256349-48-0 | 435.47 | 10mM | VEGFR;PDGFR;c-Kit;Aurora Kinase;c-Fms;FLT |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |