ATM/ATR inhibitor kit 包含ATM/ATR 抑制剂,ATM 和ATR 都是PI3K 相关激酶蛋白家族的成员,ATM 主要参与DNA 双链断裂的修复,可以在进入有丝分裂前有更多的时间进行DNA 损伤修复,也能激活相应的衰老或凋亡途径。ATR 主要参与DNA 单链断裂修复,磷酸化CDC25、CDK1和CDK2使其失活,从而阻滞G1/S 或G2/M 细胞周期进程。TargetMol 为您提供19种精选ATM/ATR 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1821 | CGK733 | 905973-89-9 | 555.84 | 10mM | ATM/ATR |
T1958 | AZ20 | 1233339-22-4 | 412.51 | 10mM | ATM/ATR; mTOR |
T2084 | ETP-46464 | 1345675-02-6 | 470.52 | 10mM | ATM/ATR; DNA-PK; mTOR; PI3K |
T2235 | Dactolisib | 915019-65-7 | 469.54 | 10mM | ATM/ATR; Autophagy; mTOR; PI3K |
T2616 | PIK-93 | 593960-11-3 | 389.88 | 10mM | ATM/ATR; Carbonic Anhydrase; DNA-PK; HSV; mTOR; PI3K; PI4K; Virus Protease |
T2669 | Berzosertib | 1232416-25-9 | 463.55 | 10mM | ATM/ATR |
T2685 | KU-55933 | 587871-26-9 | 395.49 | 10mM | ATM/ATR; Autophagy; DNA-PK; mTOR; PI3K |
T2925 | Schisandrin B | 61281-37-6 | 400.46 | 10mM | ATM/ATR; Autophagy; Reactive Oxygen Species |
T3032 | VE-821 | 1232410-49-9 | 368.41 | 10mM | ATM/ATR |
T3134 | (Z)-Mirin | 1198097-97-0 | 220.25 | 10mM | ATM/ATR |
T3338 | Ceralasertib | 1352226-88-0 | 412.51 | 10mM | ATM/ATR |
T6100 | Torin 2 | 1223001-51-1 | 432.4 | 10mM | Apoptosis; ATM/ATR; Autophagy; DNA-PK; mTOR |
T6261 | CP-466722 | 1080622-86-1 | 349.35 | 10mM | ATM/ATR |
T6283 | Wortmannin | 19545-26-7 | 428.43 | 10mM | Antibiotic; ATM/ATR; Autophagy; DNA-PK; PI3K; PLK; Serine/threonin kinase |
T6612 | NU6027 | 220036-08-8 | 251.28 | 10mM | ATM/ATR; CDK; DNA-PK |
T4443 | AZ32 | 2288709-96-4 | 328.37 | 10mM | ATM/ATR |
T5175 | azd1390 | 2089288-03-7 | 477.57 | 10mM | ATM/ATR |
T7318 | Elimusertib | 1876467-74-1 | 375.43 | 10mM | ATM/ATR |
T10468 | Elimusertib hydrochloride(1876467-74-1 free base) | T10468 | 411.89 | 10mM | ATM/ATR |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |