Androgen Receptor antagonist kit 包含雄激素受体拮抗剂,雄激素受体属于核受体超家族中的类固醇受体,与雄激素结合后,激活第二信使信号通路,调控靶基因的转录和翻译,从而影响生殖、骨骼肌、心血管、神经、免疫、造血系统的发育和稳态维持等方面。TargetMol 为您提供43种精选雄激素受体拮抗剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0272 | Nilutamide | 63612-50-0 | 317.22 | 10mM | Androgen Receptor |
T0380 | Bicalutamide | 90357-06-5 | 430.37 | 10mM | Androgen Receptor; Autophagy |
T0489 | Flutamide | 13311-84-7 | 276.21 | 10mM | Androgen Receptor |
T1167 | Cyproterone acetate | 427-51-0 | 416.94 | 10mM | Androgen Receptor |
T1541 | Drospirenone | 67392-87-4 | 366.49 | 10mM | Androgen Receptor; COX; Estrogen/progestogen Receptor; Glucocorticoid Receptor; progesterone receptor |
T1596 | Chlormadinone acetate | 302-22-7 | 404.93 | 10mM | Androgen Receptor; progesterone receptor |
T2236 | RU 58841 | 154992-24-2 | 369.34 | 10mM | Androgen Receptor |
T2339 | Apalutamide | 956104-40-8 | 477.43 | 10mM | Androgen Receptor; GABA Receptor |
T2895 | Lupeol | 545-47-1 | 426.73 | 10mM | Akt; Androgen Receptor; Apoptosis |
T2991 | 3,3'-Diindolylmethane | 1968-05-4 | 246.31 | 10mM | Androgen Receptor; Autophagy |
T3357 | Clascoterone | 19608-29-8 | 402.52 | 10mM | Androgen Receptor |
T3393 | Triptophenolide | 74285-86-2 | 312.4 | 10mM | Androgen Receptor |
T6002 | Enzalutamide | 915087-33-1 | 464.44 | 10mM | Androgen Receptor; Autophagy |
T6400 | AZD3514 | 1240299-33-5 | 519.56 | 10mM | Androgen Receptor |
T6509 | Galeterone | 851983-85-2 | 388.55 | 10mM | Androgen Receptor; P450 |
T6829 | EPI-001 | 227947-06-0 | 394.89 | 10mM | Androgen Receptor; Apoptosis; PPAR |
T6889 | MI-136 | 1628316-74-4 | 470.51 | 10mM | Androgen Receptor; Apoptosis; Epigenetic Reader Domain |
T6915 | Darolutamide | 1297538-32-9 | 398.85 | 10mM | Androgen Receptor |
T7440 | p,p'-DDE | 72-55-9 | 318 | 10mM | Androgen Receptor; Drug Metabolite |
T7690 | 2-hydroxy Flutamide | 52806-53-8 | 292.21 | 10mM | Androgen Receptor |
T8592 | CTK8A3536 | 926228-58-2 | 276.35 | 10mM | Androgen Receptor |
T13273 | UT-34 | 2168525-92-4 | 356.27 | 10mM | Androgen Receptor |
TQ0209 | Ailanthone | 981-15-7 | 376.4 | 10mM | Androgen Receptor |
TQ0214 | Dimethylcurcumin | 52328-98-0 | 396.43 | 10mM | Androgen Receptor |
T19450 | N-desmethyl Enzalutamide | 1242137-16-1 | 450.41 | 10mM | Androgen Receptor |
TCS1372 | Atraric acid | 4707-47-5 | 196.2 | 10mM | Androgen Receptor; phosphatase |
T8933 | JNJ-63576253 free base | 2110426-27-0 | 502.51 | 10mM | Androgen Receptor |
T22263 | Bavdegalutamide | 2222112-77-6 | 812.29 | 10mM | Androgen Receptor |
T12323 | ORM-15341 | 1297537-33-7 | 396.83 | 10mM | Androgen Receptor |
T14008 | 2,2,5,7,8-Pentamethyl-6-Chromanol | 950-99-2 | 220.31 | 10mM | Androgen Receptor |
T13272 | UT-155 | 2031161-35-8 | 405.35 | 10mM | Androgen Receptor |
T15445 | Proxalutamide | 1398046-21-3 | 517.5 | 10mM | Androgen Receptor; SARS-CoV |
T9246 | JNJ-63576253 | 2110428-64-1 | 538.97 | 10mM | Androgen Receptor |
T10359 | AR antagonist 1 | 1818885-54-9 | 278.78 | 10mM | Androgen Receptor; Ligand for E3 Ligase; Ligands for Target Protein for PROTAC |
T12146 | N-Desmethyl-Apalutamide | 1332391-11-3 | 463.41 | 10mM | Androgen Receptor; P450 |
T9179 | CLP-3094 | 312749-73-8 | 304.8 | 10mM | Androgen Receptor |
T14116 | ACP-105 | 899821-23-9 | 290.79 | 10mM | Androgen Receptor |
T12928 | SK33 | 1928724-23-5 | 500.31 | 10mM | Androgen Receptor |
T29111 | VPC-13566 | 218464-59-6 | 258.32 | 10mM | Androgen Receptor |
T20625 | Prochloraz | 67747-09-5 | 376.67 | 10mM | AhR; Androgen Receptor; Antifungal; Estrogen Receptor/ERR |
T24943 | VPC-14228 | 19983-28-9 | 246.33 | 10mM | Androgen Receptor |
T39695 | ARD-2128 | 2222111-87-5 | 820.38 | 10mM | Androgen Receptor |
T21740 | RD162 | 915087-27-3 | 476.45 | 10mM | Androgen Receptor |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |