AMPAR antagonist/activator kit 包含AMPA 受体拮抗剂/激活剂,AMPA 受体介导中枢神经系统快速兴奋性突触传递,诱发和维持长时程的增强和抑制,参与调节学习、记忆活动,参与谷氨酸介导的兴奋性损伤、tau 蛋白的异常磷酸化及神经原纤维缠结的形成等。AMPA 受体数目和功能异常可能导致阿尔兹海默病的发生。TargetMol 为您提供32种精选AMPA 受体拮抗剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0051 | Urethane | 51-79-6 | 89.09 | 10mM | AChR; Antibacterial; Chloride channel; GABA Receptor; GluR; NMDAR; Parasite |
T0333 | Aniracetam | 72432-10-1 | 219.24 | 10mM | 5-HT Receptor; AChR; Dopamine Receptor; GluR; iGluR |
T0426 | Piracetam | 7491-74-9 | 142.16 | 10mM | GluR; iGluR |
T1884 | CX516 | 154235-83-3 | 241.29 | 10mM | GluR; iGluR |
T3379 | Decanoic Acid | 334-48-5 | 172.26 | 10mM | GluR; iGluR |
T3473 | (S)-ATPO | 252930-37-3 | 322.25 | 10mM | GluR |
T3957 | Farampator | 211735-76-1 | 231.26 | 10mM | GluR; iGluR |
T4113 | NBQX | 118876-58-7 | 336.28 | 10mM | GluR; iGluR |
T7304 | DNQX | 2379-57-9 | 252.14 | 10mM | GluR; iGluR |
T7178 | CNQX | 115066-14-3 | 232.15 | 10mM | GluR; iGluR |
T7579 | 1-BCP | 34023-62-6 | 233.26 | 10mM | GluR; iGluR |
T7580 | CX546 | 215923-54-9 | 247.29 | 10mM | Autophagy; iGluR |
T7706 | LY-404187 | 211311-95-4 | 342.46 | 10mM | GluR; iGluR |
T7823 | IDRA-21 | 22503-72-6 | 232.68 | 10mM | GluR |
T8435 | YM90K | 154164-30-4 | 309.66 | 10mM | GluR; iGluR |
T8458 | CNQX disodium | 479347-85-8 | 276.12 | 10mM | iGluR |
T8779 | HBT1 | 489408-02-8 | 386.39 | 10mM | GluR |
T16402 | Org-26576 | 1026791-61-6 | 204.23 | 10mM | GluR; iGluR |
TP2111L | TAT-GluA2 3Y acetate(1404188-93-7 free base) | TP2111L | 2634.02 | 10mM | GluR |
T15369L | gamma-DGG acetate(6729-55-1 free base) | T15369L | 264.23 | 10mM | GluR |
TP1944L1 | pep2-SVKI acetate | TP1944L1 | 1344.51 | 10mM | GluR |
T50094 | DL-Willardiine | 19772-76-0 | 199.16 | 10mM | Others |
T16977 | Talampanel | 161832-65-1 | 337.37 | 10mM | Apoptosis; GluR |
T12406 | PEPA | 141286-78-4 | 402.44 | 10mM | iGluR |
T19698 | CX614 | 191744-13-5 | 247.25 | 10mM | GluR |
T17179 | Tulrampator | 1038984-31-4 | 380.37 | 10mM | iGluR |
T15623 | JNJ-61432059 | 2035814-50-5 | 443.47 | 10mM | iGluR |
T13480 | (S)-(-)-5-Fluorowillardiine | 140187-23-1 | 217.15 | 10mM | iGluR |
T20571 | cis-PDA | 46026-75-9 | 173.17 | 10mM | GluR; iGluR; NMDAR |
T37734 | AMPA receptor modulator-2 | 2034181-36-5 | 404.29 | 10mM | GluR |
T15820 | Mibampator | 375345-95-2 | 438.6 | 10mM | iGluR |
T27951 | LY392098 | 211311-39-6 | 335.44 | 10mM | iGluR;GluR |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |