β-/γ-secretase inhibitor kit 包含β-/γ-分泌酶抑制剂,β-secretase 是以 BACE1 为活性中心,Aph-1、Pen-2、nicastrin 的复合体;γ-secretase 是以 presenilin1 或 presenilin2 为活性中心的,与 Aph-1、Pen-2、nicastrin 组成的复合体,主要参与β-淀粉样蛋白前体(APP)和Notch 等重要跨膜蛋白的切割和水解过程。TargetMol 为您提供38种精选β-/γ-分泌酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T2262 | Itanapraced | 749269-83-8 | 325.16 | 10mM | Beta Amyloid; Gamma-secretase |
T2625 | MK-0752 | 471905-41-6 | 442.9 | 10mM | Beta Amyloid; Gamma-secretase |
T2639 | LY2811376 | 1194044-20-6 | 320.36 | 10mM | BACE; Beta Amyloid; Beta-secretase |
T3285 | Eslicarbazepine Acetate | 236395-14-5 | 296.32 | 10mM | Beta-secretase; Sodium Channel |
T3633 | Crenigacestat | 1421438-81-4 | 464.44 | 10mM | Gamma-secretase |
T3769 | Tenuifolin | 20183-47-5 | 680.37 | 10mM | AChE; Beta-secretase |
T4398 | LX2343 | 333745-53-2 | 474.91 | 10mM | Autophagy; BACE; Beta Amyloid; Beta-secretase; PI3K |
T6058 | LY2886721 | 1262036-50-9 | 390.41 | 10mM | BACE; Beta-secretase |
T6063 | LY-411575 | 209984-57-6 | 479.48 | 10mM | Apoptosis; Gamma-secretase |
T6125 | Semagacestat | 425386-60-3 | 361.44 | 10mM | Beta Amyloid; Gamma-secretase |
T6135 | YO-01027 | 209984-56-5 | 463.48 | 10mM | Gamma-secretase |
T6202 | DAPT | 208255-80-5 | 432.46 | 10mM | Apoptosis; Autophagy; Beta Amyloid; Gamma-secretase |
T6249 | Avagacestat | 1146699-66-2 | 520.88 | 10mM | Gamma-secretase |
T6274 | RO4929097 | 847925-91-1 | 469.4 | 10mM | Beta Amyloid; Gamma-secretase |
T6772 | AZD3839 free base | 1227163-84-9 | 431.41 | 10mM | BACE; Beta-secretase |
T6870 | L-685458 | 292632-98-5 | 672.85 | 10mM | Apoptosis; Gamma-secretase |
T6935 | Nirogacestat | 1290543-63-3 | 489.64 | 10mM | Apoptosis; Gamma-secretase |
T7011 | Verubecestat | 1286770-55-5 | 523.43 | 10mM | BACE; Beta-secretase |
T2S1181 | Aloenin | 38412-46-3 | 410.37 | 10mM | AChR; Beta-secretase |
T5S2361 | Epiberberine | 6873-09-2 | 336.36 | 10mM | AChE; AChR; BACE; Beta-secretase; ERK; MEK |
T8179 | Aloeresin D | 105317-67-7 | 556.6 | 10mM | BACE; Beta-secretase |
T15184 | E 2012 | 870843-42-8 | 419.49 | 10mM | Gamma-secretase |
T9015 | LY900009 | 209984-68-9 | 409.49 | 10mM | Gamma-secretase |
T16294 | NGP555 | 1304630-27-0 | 406.52 | 10mM | Gamma-secretase |
T11175 | Elenbecestat | 1388651-30-6 | 437.44 | 10mM | BACE; Beta-secretase |
T22678 | 3,5-Bis(4-nitrophenoxy)benzoic acid | 173550-33-9 | 396.31 | 10mM | Gamma-secretase |
T21890 | JLK6 | 62252-26-0 | 225.63 | 10mM | Gamma-secretase |
T9422 | Fosciclopirox | 1380539-06-9 | 317.27 | 10mM | Gamma-secretase |
T16133 | MRK-560 | 677772-84-8 | 517.92 | 10mM | Gamma-secretase |
T3285L | Eslicarbazepine | 104746-04-5 | 254.28 | 10mM | Beta-secretase; sodium channel |
T11358 | gamma-secretase modulator 1 | 1172637-87-4 | 416.54 | 10mM | Gamma-secretase |
T11178L | ELN318463 racemate | 851599-82-1 | 471.8 | 10mM | Gamma-secretase |
T2759 | Loganin | 18524-94-2 | 390.38 | 10mM | AChE; AChR; Apoptosis; BACE; NF-κB |
T3394 | Timosaponin BII | 136656-07-0 | 920.07 | 10mM | BACE; Beta Amyloid |
TN1343 | 8-Geranyloxypsoralen | 7437-55-0 | 338.4 | 10mM | Anti-infection; BACE; P450 |
T3161L | BACE-IN-1 acetate | T3161L | 1711.86 | 10mM | BACE |
T12188 | NB-360 | 1262857-73-7 | 449.4 | 10mM | BACE |
T13253 | Umibecestat | 1387560-01-1 | 513.8 | 10mM | BACE |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |